Table of Contents

Articles

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- MICHIHISA MIYAKE and
- SHOJI SHIBATA
A Novel Mode of Neurotoxin Action: A Polypeptide Toxin Isolated from Anemonia sulcata Shifts the Voltage Dependence of the Maximal Rate of Rise of Na⁺ Action Potentials in a Mouse Neuronal Clone
Mol Pharmacol November 1981 20:453-456; doi:
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- MARGARET A. CASCIERI,
- MARVIN M. GOLDENBERG,
- and TEHMING LIANG
Biological Activity of Substance P Methyl Ester
Mol Pharmacol November 1981 20:457-459; doi:
- Abstract
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- PAULA H. STERN,
- YOKO TANAKA,
- HECTOR F. DELUCA,
- NOBUO IKEKAWA,
- and YOSHIRO KOBAYASHI
Bone Resorptive Activity of Side-Chain Fluoro Derivatives of 25-Hydroxy- and 1α,25-Dihydroxyvitamin D₃ in Culture
Mol Pharmacol November 1981 20:460-462; doi:
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- VINCENT HOMBURGER,
- MARGUERITE LUCAS,
- ETELKA ROSENBAUM,
- GÉRARD VASSENT,
- and JOËL BOCKAERT
Presence of Both Beta₁- and Beta₂-Adrenergic Receptors in a Single Cell Type
Mol Pharmacol November 1981 20:463-469; doi:
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- TOMMASO COSTA,
- LAURA RUSSELL,
- CANDACE B. PERT,
- and DAVID RODBARD
Halide- and γ-Aminobutyric Acid-Induced Enhancement of Diazepam Receptors in Rat Brain: Reversal by Disulfonic Stilbene Blockers of Anion Channels
Mol Pharmacol November 1981 20:470-476; doi:
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- JOHN W. REGAN,
- WILLIAM R. ROESKE,
- JEFFREY B. MALICK,
- SUSAN H. YAMAMURA,
- and HENRY I. YAMAMURA
γ-Aminobutyric Acid Enhancement of CL 218,872 Affinity and Evidence of Benzodiazepine Receptor Heterogeneity
Mol Pharmacol November 1981 20:477-483; doi:
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- MARIE-CLAUDE FOURNIE-ZALUSKI,
- GILLES GACEL,
- BERNARD MAIGRET,
- SAMUEL PREMILAT,
- and BERNARD P. ROQUES
Structural Requirements for Specific Recognition of µ or δ Opiate Receptors
Mol Pharmacol November 1981 20:484-491; doi:
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- ANWAR-SAAD A. ABD-ELFATTAH and
- ADIL E. SHAMOO
Regeneration of a Functionally Active Rat Brain Muscarinic Receptor by D-Penicillamine after Inhibition with Methylmercury and Mercuric Chloride: Evidence for Essential Sulfhydryl Groups in Muscarinic Receptor Binding Sites
Mol Pharmacol November 1981 20:492-497; doi:
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- ANTHONY P. YOUNG and
- DAVID S. SIGMAN
Allosteric Effects of Volatile Anesthetics on the Membrane-Bound Acetylcholine Receptor Protein: I. Stabilization of the High-Affinity State
Mol Pharmacol November 1981 20:498-505; doi:
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- ANTHONY P. YOUNG,
- JANIS R. OSHIKI,
- and DAVID S. SIGMAN
Allosteric Effects of Volatile Anesthetics on the Membrane-Bound Acetylcholine Receptor Protein: II. Alteration of α-Bungarotoxin Binding Kinetics
Mol Pharmacol November 1981 20:506-510; doi:
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- N. SHAKER,
- A. T. ELDEFRAWI,
- E. R. MILLER,
- and M. E. ELDEFRAWI
Interaction of Tricyclic Antidepressants with the Ionic Channel of the Acetylcholine Receptor of Torpedo Electric Organ
Mol Pharmacol November 1981 20:511-518; doi:
- Abstract
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- ESAM EL-FAKAHANY and
- ELLIOTT RICHELSON
Phenoxybenzamine and Dibenamine Interactions with Calcium Channel Effectors of the Muscarinic Receptor
Mol Pharmacol November 1981 20:519-525; doi:
- Abstract
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- WILLIAM A. CATTERALL and
- JEFFREY COPPERSMITH
High-Affinity Saxitoxin Receptor Sites in Vertebrate Heart: Evidence for Sites Associated with Autonomic Nerve Endings
Mol Pharmacol November 1981 20:526-532; doi:
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- WILLIAM A. CATTERALL and
- JEFFREY COPPERSMITH
Pharmacological Properties of Sodium Channels in Cultured Rat Heart Cells
Mol Pharmacol November 1981 20:533-542; doi:
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- KLAUS TURNHEIM,
- ANTON LUGER,
- and MARKUS GRASL
Kinetic Analysis of the Amiloride-Sodium Entry Site Interaction in Rabbit Colon
Mol Pharmacol November 1981 20:543-550; doi:
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- MARTIN WEHLING,
- ARNOLD SCHWARTZ,
- KYRA WHITMER,
- GUNTER GRUPP,
- INGRID L. GRUPP,
- and EARL T. WALLICK
Interaction of Chlormadinone Acetate with the Ouabain Binding Site of Na⁺, K⁺-ATPase
Mol Pharmacol November 1981 20:551-557; doi:
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- GIULIANO BANDOLI,
- DORE A. CLEMENTE,
- ANTONIO GRASSI,
- and GIUSEPPE C. PAPPALARDO
Molecular Determinants for Drug-Receptor Interactions: 1. Solid-State Structure and Conformation of the Novel Nootropic Agent 2-Pyrrolidone-N-Acetamide: X-Ray and Theoretical SCF-MO Studies
Mol Pharmacol November 1981 20:558-564; doi:
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- RONALD L. GOLDBERG,
- TOMMASO COSTA,
- WILLIAM H. HABIG,
- LEONARD D. KOHN,
- and M. CAROLYN HARDEGREE
Characterization of Fragment C and Tetanus Toxin Binding to Rat Brain Membranes
Mol Pharmacol November 1981 20:565-570; doi:
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- HIROYOSHI HIDAKA,
- MASAHISA ASANO,
- and TOSHIO TANAKA
Activity-Structure Relationship of Calmodulin Antagonists: Naphthalenesulfonamide Derivatives
Mol Pharmacol November 1981 20:571-578; doi:
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- H. HAMBOECK,
- R. W. FISCHER,
- E. E. DI IORIO,
- and K. H. WINTERHALTER
The Binding of s-Triazine Metabolites to Rodent Hemoglobins Appears Irrelevant to Other Species
Mol Pharmacol November 1981 20:579-584; doi:
- Abstract
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- JAMES G. KENIMER and
- MARSHALL NIRENBERG
Desensitization of Adenylate Cyclase to Prostaglandin E₁ or 2-Chloroadenosine
Mol Pharmacol November 1981 20:585-591; doi:
- Abstract
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- SAM WEISS and
- GEORGE I. DRUMMOND
Dopamine- and Serotonin-Sensitive Adenylate Cyclase in the Gill of Aplysia californica
Mol Pharmacol November 1981 20:592-597; doi:
- Abstract
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- JEAN-PIERRE HÉNICHART,
- RAYMOND HOUSSIN,
- CAROLE GORS,
- and FRANÇOIS BAERT
Conformational Analysis of a New Analgesic Triazolinethione: Structural Comparisons with Antipyrine
Mol Pharmacol November 1981 20:598-601; doi:
- Abstract
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- LIBBY M. YUNGER and
- RICHARD D. CRAMER III
Measurement and Correlation of Partition Coefficients of Polar Amino Acids
Mol Pharmacol November 1981 20:602-608; doi:
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- S. HANDWERGER,
- J. BARRETT,
- S. BARRY,
- E. MARKOFF,
- P. ZEITLER,
- B. CWIKEL,
- and M. SIEGEL
Stimulation of Human Placental Lactogen Release by Arachidonic Acid
Mol Pharmacol November 1981 20:609-613; doi:
- Abstract
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- STEVEN J. WHITE and
- ROBERT S. JACOBS
Inhibition of Cell Division and of Microtubule Assembly by Elatone, a Halogenated Sesquiterpene
Mol Pharmacol November 1981 20:614-620; doi:
- Abstract
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- VALENTINE DURUIBE and
- GOPI A. TEJWANI
The Effect of Ethanol on the Activities of the Key Gluconeogenic and Glycolytic Enzymes of Rat Liver
Mol Pharmacol November 1981 20:621-630; doi:
- Abstract
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- JON-SVERRE SCHANCHE,
- TONE SCHANCHE,
- and PER MAGNE UELAND
Inhibition of Phospholipid Methyltransferase(s) from Rat Liver Plasma Membranes by Analogues of S-Adenosylhomocysteine
Mol Pharmacol November 1981 20:631-636; doi:
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- MICHAEL HAMRELL,
- JOHN LASZLO,
- OLIVER E. BROWN,
- and W. DAVID SEDWICK
Toxicity of Methotrexate and Metoprine in a Dihydrofolate Reductase Gene-Amplified Mouse Cell Line
Mol Pharmacol November 1981 20:637-643; doi:
- Abstract
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- HSIN-LI LIN and
- ROBERT I. GLAZER
The Comparative Effects of 5-Azacytidine and Dihydro-5-azacytidine on Polysomal RNA in Ehrlich Ascites Cells in Vitro
Mol Pharmacol November 1981 20:644-648; doi:
- Abstract
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- ZONG-RU GUO,
- STEPHEN W. DIETRICH,
- CORWIN HANSCH,
- BRUICE J. DOLNICK,
- and JOSEPH R. BERTINO
A Comparison of the Inhibition of Bovine and Murine Leukemia Dihydrofolate Reductase by 4,6-Diamino-1,2-dihydro-2,2-dimethyl-1-(3-X-phenyl)-s-Triazines
Mol Pharmacol November 1981 20:649-656; doi:
- Abstract
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- ROBERT I. GLAZER and
- KATHLEEN D. HARTMAN
Cytokinetic and Biochemical Effects of Sangivamycin in Human Colon Carcinoma Cells in Culture
Mol Pharmacol November 1981 20:657-661; doi:
- Abstract
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- IAIN G. C. ROBERTSON,
- RICHARD M. PHILPOT,
- ERROL ZEIGER,
- and C. ROLAND WOLF
Specificity of Rabbit Pulmonary Cytochrome P-450 Isozymes in the Activation of Several Aromatic Amines and Aflatoxin B₁
Mol Pharmacol November 1981 20:662-668; doi:
- Abstract
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- JORDAN L. HOLTZMAN,
- DAUNE L. CRANKSHAW,
- FRANCIS J. PETERSON,
- and CARL F. POLNASZEK
The Kinetics of the Aerobic Reduction of Nitrofurantoin by NADPH-Cytochrome P-450 (c) Reductase
Mol Pharmacol November 1981 20:669-673; doi:
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- DAVID CHOU,
- CARL F. POLNASZEK,
- YUL YOST,
- ILO E. LEPPIK,
- and JORDAN L. HOLTZMAN
Application of Spin Labeling to Drug Assays: II. Determination of the Binding of [¹⁴C]-Phenytoin and Spin-Labeled Phenytoins to Albumin and Human Serum
Mol Pharmacol November 1981 20:674-680; doi:
- Abstract
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- GURMIT SINGH and
- KENNETH W. RENTON
Interferon-Mediated Depression of Cytochrome P-450-Dependent Drug Biotransformation
Mol Pharmacol November 1981 20:681-684; doi:
- Abstract
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- DAVID E. MOODY,
- JACQUELINE L. JAMES,
- GARY A. CLAWSON,
- and EDWARD A. SMUCKLER
Correlations among the Changes in Hepatic Microsomal Components after Intoxication with Alkyl Halides and Other Hepatotoxins
Mol Pharmacol November 1981 20:685-693; doi:
- Abstract
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- THOMAS H. HUDSON and
- GARY L. JOHNSON
Functional Alterations in Components of Pigeon Erythrocyte Adenylate Cyclase following Desensitization to Isoproterenol
Mol Pharmacol November 1981 20:694-703; doi:
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- YASUNORI KANAHO,
- TAKASHI SATO,
- and TATSUZO FUJII
The Affinity of Various Phenothiazine Drugs for Membranes of Intact Human Erythrocytes and Their Membrane-Transforming Activity
Mol Pharmacol November 1981 20:704-708; doi:
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- THOMAS T. KAWABATA,
- F. PETER GUENGERICH,
- and JEFFREY BARON
An Immunohistochemical Study on the Localization and Distribution of Epoxide Hydrolase within Livers of Untreated Rats
Mol Pharmacol November 1981 20:709-714; doi:
- Abstract
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Articles

A Novel Mode of Neurotoxin Action: A Polypeptide Toxin Isolated from Anemonia sulcata Shifts the Voltage Dependence of the Maximal Rate of Rise of Na+ Action Potentials in a Mouse Neuronal Clone

Biological Activity of Substance P Methyl Ester

Bone Resorptive Activity of Side-Chain Fluoro Derivatives of 25-Hydroxy- and 1α,25-Dihydroxyvitamin D3 in Culture

Presence of Both Beta1- and Beta2-Adrenergic Receptors in a Single Cell Type

Halide- and γ-Aminobutyric Acid-Induced Enhancement of Diazepam Receptors in Rat Brain: Reversal by Disulfonic Stilbene Blockers of Anion Channels

γ-Aminobutyric Acid Enhancement of CL 218,872 Affinity and Evidence of Benzodiazepine Receptor Heterogeneity

Structural Requirements for Specific Recognition of µ or δ Opiate Receptors

Regeneration of a Functionally Active Rat Brain Muscarinic Receptor by D-Penicillamine after Inhibition with Methylmercury and Mercuric Chloride: Evidence for Essential Sulfhydryl Groups in Muscarinic Receptor Binding Sites

Allosteric Effects of Volatile Anesthetics on the Membrane-Bound Acetylcholine Receptor Protein: I. Stabilization of the High-Affinity State

Allosteric Effects of Volatile Anesthetics on the Membrane-Bound Acetylcholine Receptor Protein: II. Alteration of α-Bungarotoxin Binding Kinetics

Interaction of Tricyclic Antidepressants with the Ionic Channel of the Acetylcholine Receptor of Torpedo Electric Organ

Phenoxybenzamine and Dibenamine Interactions with Calcium Channel Effectors of the Muscarinic Receptor

High-Affinity Saxitoxin Receptor Sites in Vertebrate Heart: Evidence for Sites Associated with Autonomic Nerve Endings

Pharmacological Properties of Sodium Channels in Cultured Rat Heart Cells

Kinetic Analysis of the Amiloride-Sodium Entry Site Interaction in Rabbit Colon

Interaction of Chlormadinone Acetate with the Ouabain Binding Site of Na+, K+-ATPase

Molecular Determinants for Drug-Receptor Interactions: 1. Solid-State Structure and Conformation of the Novel Nootropic Agent 2-Pyrrolidone-N-Acetamide: X-Ray and Theoretical SCF-MO Studies

Characterization of Fragment C and Tetanus Toxin Binding to Rat Brain Membranes

Activity-Structure Relationship of Calmodulin Antagonists: Naphthalenesulfonamide Derivatives

The Binding of s-Triazine Metabolites to Rodent Hemoglobins Appears Irrelevant to Other Species

Desensitization of Adenylate Cyclase to Prostaglandin E1 or 2-Chloroadenosine

Dopamine- and Serotonin-Sensitive Adenylate Cyclase in the Gill of Aplysia californica

Conformational Analysis of a New Analgesic Triazolinethione: Structural Comparisons with Antipyrine

Measurement and Correlation of Partition Coefficients of Polar Amino Acids

Stimulation of Human Placental Lactogen Release by Arachidonic Acid

Inhibition of Cell Division and of Microtubule Assembly by Elatone, a Halogenated Sesquiterpene

The Effect of Ethanol on the Activities of the Key Gluconeogenic and Glycolytic Enzymes of Rat Liver

Inhibition of Phospholipid Methyltransferase(s) from Rat Liver Plasma Membranes by Analogues of S-Adenosylhomocysteine

Toxicity of Methotrexate and Metoprine in a Dihydrofolate Reductase Gene-Amplified Mouse Cell Line

The Comparative Effects of 5-Azacytidine and Dihydro-5-azacytidine on Polysomal RNA in Ehrlich Ascites Cells in Vitro

A Comparison of the Inhibition of Bovine and Murine Leukemia Dihydrofolate Reductase by 4,6-Diamino-1,2-dihydro-2,2-dimethyl-1-(3-X-phenyl)-s-Triazines

Cytokinetic and Biochemical Effects of Sangivamycin in Human Colon Carcinoma Cells in Culture

Specificity of Rabbit Pulmonary Cytochrome P-450 Isozymes in the Activation of Several Aromatic Amines and Aflatoxin B1

The Kinetics of the Aerobic Reduction of Nitrofurantoin by NADPH-Cytochrome P-450 (c) Reductase

Application of Spin Labeling to Drug Assays: II. Determination of the Binding of [14C]-Phenytoin and Spin-Labeled Phenytoins to Albumin and Human Serum

Interferon-Mediated Depression of Cytochrome P-450-Dependent Drug Biotransformation

Correlations among the Changes in Hepatic Microsomal Components after Intoxication with Alkyl Halides and Other Hepatotoxins

Functional Alterations in Components of Pigeon Erythrocyte Adenylate Cyclase following Desensitization to Isoproterenol

The Affinity of Various Phenothiazine Drugs for Membranes of Intact Human Erythrocytes and Their Membrane-Transforming Activity

An Immunohistochemical Study on the Localization and Distribution of Epoxide Hydrolase within Livers of Untreated Rats

This Issue

Current Issue

A Novel Mode of Neurotoxin Action: A Polypeptide Toxin Isolated from Anemonia sulcata Shifts the Voltage Dependence of the Maximal Rate of Rise of Na⁺ Action Potentials in a Mouse Neuronal Clone

Bone Resorptive Activity of Side-Chain Fluoro Derivatives of 25-Hydroxy- and 1α,25-Dihydroxyvitamin D₃ in Culture

Presence of Both Beta₁- and Beta₂-Adrenergic Receptors in a Single Cell Type

Interaction of Chlormadinone Acetate with the Ouabain Binding Site of Na⁺, K⁺-ATPase

Desensitization of Adenylate Cyclase to Prostaglandin E₁ or 2-Chloroadenosine

Specificity of Rabbit Pulmonary Cytochrome P-450 Isozymes in the Activation of Several Aromatic Amines and Aflatoxin B₁

Application of Spin Labeling to Drug Assays: II. Determination of the Binding of [¹⁴C]-Phenytoin and Spin-Labeled Phenytoins to Albumin and Human Serum