Table of Contents

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- J Lerma and
- R Martín del Río
Chloride transport blockers prevent N-methyl-D-aspartate receptor-channel complex activation.
Mol Pharmacol February 1992 41:217-222
- Abstract
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- W Y Gao,
- F S Han,
- C Storm,
- W Egan,
- and Y C Cheng
Phosphorothioate oligonucleotides are inhibitors of human DNA polymerases and RNase H: implications for antisense technology.
Mol Pharmacol February 1992 41:223-229
- Abstract
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- A J Townsend,
- C P Tu,
- and K H Cowan
Expression of human mu or alpha class glutathione S-transferases in stably transfected human MCF-7 breast cancer cells: effect on cellular sensitivity to cytotoxic agents.
Mol Pharmacol February 1992 41:230-236
- Abstract
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- X B Kong,
- L Rubin,
- L I Chen,
- G Ciszewska,
- K A Watanabe,
- W P Tong,
- F M Sirotnak,
- and T C Chou
Topoisomerase II-mediated DNA cleavage activity and irreversibility of cleavable complex formation induced by DNA intercalator with alkylating capability.
Mol Pharmacol February 1992 41:237-244
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- W B Parker,
- S C Shaddix,
- P W Allan,
- G Arnett,
- L M Rose,
- W M Shannon,
- Y F Shealy,
- J A Montgomery,
- J A Secrist, 3rd,
- and L L Bennett, Jr
Incorporation of the carbocyclic analog of 2'-deoxyguanosine into the DNA of herpes simplex virus and of HEp-2 cells infected with herpes simplex virus.
Mol Pharmacol February 1992 41:245-251
- Abstract
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- D A Weidner,
- E G Bridges,
- E M Cretton,
- and J P Sommadossi
Comparative effects of 3'-azido-3'-deoxythymidine and its metabolite 3'-amino-3'-deoxythymidine on hemoglobin synthesis in K-562 human leukemia cells.
Mol Pharmacol February 1992 41:252-258
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- R Hyland,
- A Gescher,
- K Thummel,
- C Schiller,
- P Jheeta,
- K Mynett,
- A W Smith,
- and J Mráz
Metabolic oxidation and toxification of N-methylformamide catalyzed by the cytochrome P450 isoenzyme CYP2E1.
Mol Pharmacol February 1992 41:259-266
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- J A Mancini,
- P Prasit,
- M G Coppolino,
- P Charleson,
- S Leger,
- J F Evans,
- J W Gillard,
- and P J Vickers
5-Lipoxygenase-activating protein is the target of a novel hybrid of two classes of leukotriene biosynthesis inhibitors.
Mol Pharmacol February 1992 41:267-272
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- B Rouot,
- N Charpentier,
- C Chabbert,
- J Carrette,
- R Zumbihl,
- J Bockaert,
- and V Homburger
Specific antibodies against Go isoforms reveal the early expression of the Go2 alpha subunit and appearance of Go1 alpha during neuronal differentiation.
Mol Pharmacol February 1992 41:273-280
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- T L Yue,
- J M Stadel,
- H M Sarau,
- E Friedman,
- J L Gu,
- D A Powers,
- M M Gleason,
- G Feuerstein,
- and H Y Wang
Platelet-activating factor stimulates phosphoinositide turnover in neurohybrid NCB-20 cells: involvement of pertussis toxin-sensitive guanine nucleotide-binding proteins and inhibition by protein kinase C.
Mol Pharmacol February 1992 41:281-289
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- K Tsutsumi and
- J M Saavedra
Heterogeneity of angiotensin II AT2 receptors in the rat brain.
Mol Pharmacol February 1992 41:290-297
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- H G Knaus,
- J Striessnig,
- S Hering,
- S Marrer,
- E Schwenner,
- H D Höltje,
- and H Glossmann
[35S]sadopine, a novel high affinity, high specific activity, L-type Ca2+ channel probe: characterization of two equipotent diastereomers with opposite allosteric properties.
Mol Pharmacol February 1992 41:298-307
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- S W Leslie,
- L M Brown,
- R D Trent,
- Y H Lee,
- J L Morris,
- T W Jones,
- P K Randall,
- S S Lau,
- and T J Monks
Stimulation of N-methyl-D-aspartate receptor-mediated calcium entry into dissociated neurons by reduced and oxidized glutathione.
Mol Pharmacol February 1992 41:308-314
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- R P Mason,
- D M Moisey,
- and L Shajenko
Cholesterol alters the binding of Ca2+ channel blockers to the membrane lipid bilayer.
Mol Pharmacol February 1992 41:315-321
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- J Snyders,
- K M Knoth,
- S L Roberds,
- and M M Tamkun
Time-, voltage-, and state-dependent block by quinidine of a cloned human cardiac potassium channel.
Mol Pharmacol February 1992 41:322-330
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- C F Valenzuela,
- J A Kerr,
- P Duvvuri,
- and D A Johnson
Modulation of phencyclidine-sensitive ethidium binding to the Torpedo acetylcholine receptor: interaction of noncompetitive inhibitors with carbamylcholine and cobra alpha-toxin.
Mol Pharmacol February 1992 41:331-336
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- J C Randle,
- T Guet,
- C Bobichon,
- C Moreau,
- P Curutchet,
- B Lambolez,
- L P de Carvalho,
- A Cordi,
- and J M Lepagnol
Quinoxaline derivatives: structure-activity relationships and physiological implications of inhibition of N-methyl-D-aspartate and non-N-methyl-D-aspartate receptor-mediated currents and synaptic potentials.
Mol Pharmacol February 1992 41:337-345
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- H Ouadid,
- J Seguin,
- A Dumuis,
- J Bockaert,
- and J Nargeot
Serotonin increases calcium current in human atrial myocytes via the newly described 5-hydroxytryptamine4 receptors.
Mol Pharmacol February 1992 41:346-351
- Abstract
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- I Hide,
- W L Padgett,
- K A Jacobson,
- and J W Daly
A2A adenosine receptors from rat striatum and rat pheochromocytoma PC12 cells: characterization with radioligand binding and by activation of adenylate cyclase.
Mol Pharmacol February 1992 41:352-359
- Abstract
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- A Laurenza,
- J D Robbins,
- and K B Seamon
Interaction of aminoalkylcarbamates of forskolin with adenylyl cyclase: synthesis of an iodinated derivative of forskolin with high affinity for adenylyl cyclase.
Mol Pharmacol February 1992 41:360-368
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- J Wess,
- D Gdula,
- and M R Brann
Structural basis of the subtype selectivity of muscarinic antagonists: a study with chimeric m2/m5 muscarinic receptors.
Mol Pharmacol February 1992 41:369-374
- Abstract
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- J B Kurz and
- J P Perkins
Isoproterenol-initiated beta-adrenergic receptor diacytosis in cultured cells.
Mol Pharmacol February 1992 41:375-381
- Abstract
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- M H Werner,
- A E Bielawska,
- and Y A Hannun
Quantitative analysis of diacylglycerol second messengers in human platelets: correlation with aggregation and secretion.
Mol Pharmacol February 1992 41:382-386
- Abstract
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- N E Ward and
- C A O'Brian
Kinetic analysis of protein kinase C inhibition by staurosporine: evidence that inhibition entails inhibitor binding at a conserved region of the catalytic domain but not competition with substrates.
Mol Pharmacol February 1992 41:387-392
- Abstract
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- R F Kletzien,
- S D Clarke,
- and R G Ulrich
Enhancement of adipocyte differentiation by an insulin-sensitizing agent.
Mol Pharmacol February 1992 41:393-398
- Abstract
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- T D Warner,
- J A Mitchell,
- P D'Orleans-Juste,
- K Ishii,
- U Förstermann,
- and F Murad
Characterization of endothelin-converting enzyme from endothelial cells and rat brain: detection of the formation of biologically active endothelin-1 by rapid bioassay.
Mol Pharmacol February 1992 41:399-403
- Abstract
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- M K Bijsterbosch and
- T J Van Berkel
Lactosylated high density lipoprotein: a potential carrier for the site-specific delivery of drugs to parenchymal liver cells.
Mol Pharmacol February 1992 41:404-411
- Abstract
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- H A Berman and
- K Leonard
Interaction of tetrahydroaminoacridine with acetylcholinesterase and butyrylcholinesterase.
Mol Pharmacol February 1992 41:412-418
- Abstract
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- T H Maren
Direct measurements of the rate constants of sulfonamides with carbonic anhydrase.
Mol Pharmacol February 1992 41:419-426
- Abstract
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- E S Roberts,
- A D Vaz,
- and M J Coon
Role of isozymes of rabbit microsomal cytochrome P-450 in the metabolism of retinoic acid, retinol, and retinal.
Mol Pharmacol February 1992 41:427-433
- Abstract
- Full Text (PDF)

Chloride transport blockers prevent N-methyl-D-aspartate receptor-channel complex activation.

Phosphorothioate oligonucleotides are inhibitors of human DNA polymerases and RNase H: implications for antisense technology.

Expression of human mu or alpha class glutathione S-transferases in stably transfected human MCF-7 breast cancer cells: effect on cellular sensitivity to cytotoxic agents.

Topoisomerase II-mediated DNA cleavage activity and irreversibility of cleavable complex formation induced by DNA intercalator with alkylating capability.

Incorporation of the carbocyclic analog of 2'-deoxyguanosine into the DNA of herpes simplex virus and of HEp-2 cells infected with herpes simplex virus.

Comparative effects of 3'-azido-3'-deoxythymidine and its metabolite 3'-amino-3'-deoxythymidine on hemoglobin synthesis in K-562 human leukemia cells.

Metabolic oxidation and toxification of N-methylformamide catalyzed by the cytochrome P450 isoenzyme CYP2E1.

5-Lipoxygenase-activating protein is the target of a novel hybrid of two classes of leukotriene biosynthesis inhibitors.

Specific antibodies against Go isoforms reveal the early expression of the Go2 alpha subunit and appearance of Go1 alpha during neuronal differentiation.

Platelet-activating factor stimulates phosphoinositide turnover in neurohybrid NCB-20 cells: involvement of pertussis toxin-sensitive guanine nucleotide-binding proteins and inhibition by protein kinase C.

Heterogeneity of angiotensin II AT2 receptors in the rat brain.

[35S]sadopine, a novel high affinity, high specific activity, L-type Ca2+ channel probe: characterization of two equipotent diastereomers with opposite allosteric properties.

Stimulation of N-methyl-D-aspartate receptor-mediated calcium entry into dissociated neurons by reduced and oxidized glutathione.

Cholesterol alters the binding of Ca2+ channel blockers to the membrane lipid bilayer.

Time-, voltage-, and state-dependent block by quinidine of a cloned human cardiac potassium channel.

Modulation of phencyclidine-sensitive ethidium binding to the Torpedo acetylcholine receptor: interaction of noncompetitive inhibitors with carbamylcholine and cobra alpha-toxin.

Quinoxaline derivatives: structure-activity relationships and physiological implications of inhibition of N-methyl-D-aspartate and non-N-methyl-D-aspartate receptor-mediated currents and synaptic potentials.

Serotonin increases calcium current in human atrial myocytes via the newly described 5-hydroxytryptamine4 receptors.

A2A adenosine receptors from rat striatum and rat pheochromocytoma PC12 cells: characterization with radioligand binding and by activation of adenylate cyclase.

Interaction of aminoalkylcarbamates of forskolin with adenylyl cyclase: synthesis of an iodinated derivative of forskolin with high affinity for adenylyl cyclase.

Structural basis of the subtype selectivity of muscarinic antagonists: a study with chimeric m2/m5 muscarinic receptors.

Isoproterenol-initiated beta-adrenergic receptor diacytosis in cultured cells.

Quantitative analysis of diacylglycerol second messengers in human platelets: correlation with aggregation and secretion.

Kinetic analysis of protein kinase C inhibition by staurosporine: evidence that inhibition entails inhibitor binding at a conserved region of the catalytic domain but not competition with substrates.

Enhancement of adipocyte differentiation by an insulin-sensitizing agent.

Characterization of endothelin-converting enzyme from endothelial cells and rat brain: detection of the formation of biologically active endothelin-1 by rapid bioassay.

Lactosylated high density lipoprotein: a potential carrier for the site-specific delivery of drugs to parenchymal liver cells.

Interaction of tetrahydroaminoacridine with acetylcholinesterase and butyrylcholinesterase.

Direct measurements of the rate constants of sulfonamides with carbonic anhydrase.

Role of isozymes of rabbit microsomal cytochrome P-450 in the metabolism of retinoic acid, retinol, and retinal.

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