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Molecular Pharmacology

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Table of Contents

March 01, 2000; Volume 57,Issue 3

Articles

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    Ca2+ Requirement for High-Affinity γ-Aminobutyric Acid (GABA) Binding at GABAB Receptors: Involvement of Serine 269 of the GABABR1 Subunit
    Thierry Galvez, Stephan Urwyler, Laurent Prézeau, Johannes Mosbacher, Cécile Joly, Barbara Malitschek, Jakob Heid, Isabelle Brabet, Wolfgang Froestl, Bernhard Bettler, Klemens Kaupmann and Jean-Philippe Pin
    Molecular Pharmacology March 2000, 57 (3) 419-426; DOI: https://doi.org/10.1124/mol.57.3.419
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    Structure-Activity Relationship of Staurosporine Analogs in Regulating Expression of Endothelial Nitric-Oxide Synthase Gene
    Huige Li and Ulrich Förstermann
    Molecular Pharmacology March 2000, 57 (3) 427-435; DOI: https://doi.org/10.1124/mol.57.3.427
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    Allosteric Interactions between the Antagonist Prazosin and Amiloride Analogs at the Human α1A-Adrenergic Receptor
    Ray A. Leppik, Anita Mynett, Sebastian Lazareno and Nigel J. M. Birdsall
    Molecular Pharmacology March 2000, 57 (3) 436-445; DOI: https://doi.org/10.1124/mol.57.3.436
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    Modulation of Dopamine D2 Receptor Signaling by Actin-Binding Protein (ABP-280)
    M. Li, J. C. Bermak, Z. W. Wang and Q. Y. Zhou
    Molecular Pharmacology March 2000, 57 (3) 446-452; DOI: https://doi.org/10.1124/mol.57.3.446
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    Characterization of Protein Kinase chk1 Essential for the Cell Cycle Checkpoint after Exposure of Human Head and Neck Carcinoma A253 Cells to a Novel Topoisomerase I Inhibitor BNP1350
    Ming-Biao Yin, Bin Guo, Udo Vanhoefer, Rami G. Azrak, Hans Minderman, Cheryl Frank, Carol Wrzosek, Harry K. Slocum and Youcef M. Rustum
    Molecular Pharmacology March 2000, 57 (3) 453-459; DOI: https://doi.org/10.1124/mol.57.3.453
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    Specific Regulation of RGS2 Messenger RNA by Angiotensin II in Cultured Vascular Smooth Muscle Cells
    Sharon L. Grant, Bernard Lassègue, Kathy K. Griendling, Masuko Ushio-Fukai, P. Reid Lyons and R. Wayne Alexander
    Molecular Pharmacology March 2000, 57 (3) 460-467; DOI: https://doi.org/10.1124/mol.57.3.460
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    Substrate-Dependent Regulation of Human ArylamineN-Acetyltransferase-1 in Cultured Cells
    Neville J. Butcher, Kenneth F. Ilett and Rodney F. Minchin
    Molecular Pharmacology March 2000, 57 (3) 468-473; DOI: https://doi.org/10.1124/mol.57.3.468
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    A Single Glycine Residue at the Entrance to the First Membrane-Spanning Domain of the γ-Aminobutyric Acid Type A Receptor β2 Subunit Affects Allosteric Sensitivity to GABA and Anesthetics
    Berit X. Carlson, A. Christine Engblom, Uffe Kristiansen, Arne Schousboe and Richard W. Olsen
    Molecular Pharmacology March 2000, 57 (3) 474-484; DOI: https://doi.org/10.1124/mol.57.3.474
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    Inhibition of c-myc Expression in Cells by Targeting an RNA-Protein Interaction Using Antisense Oligonucleotides
    Christopher M. Coulis, Chunja Lee, Violet Nardone and Rebecca D. Prokipcak
    Molecular Pharmacology March 2000, 57 (3) 485-494; DOI: https://doi.org/10.1124/mol.57.3.485
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    Functional Inactivation of the Nociceptin Receptor by Alanine Substitution of Glutamine 286 at the C Terminus of Transmembrane Segment VI: Evidence from a Site-Directed Mutagenesis Study of the ORL1 Receptor Transmembrane-Binding Domain
    Lionel Mouledous, Christopher M. Topham, Christiane Moisand, Catherine Mollereau and Jean-Claude Meunier
    Molecular Pharmacology March 2000, 57 (3) 495-502; DOI: https://doi.org/10.1124/mol.57.3.495
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    Effect of p53 Status on Sensitivity to Platinum Complexes in a Human Ovarian Cancer Cell Line
    Katharine E. Pestell, Stephen M. Hobbs, Jenny C. Titley, Lloyd R. Kelland and Michael I. Walton
    Molecular Pharmacology March 2000, 57 (3) 503-511; DOI: https://doi.org/10.1124/mol.57.3.503
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    Hematotoxicity of the Chinese Herbal Medicine Tripterygium wilfordii Hook f in CD34-Positive Human Bone Marrow Cells
    David W. Pyatt, Yanzhu Yang, Brenda Mehos, Anh Le, Wayne Stillman and Richard D. Irons
    Molecular Pharmacology March 2000, 57 (3) 512-518; DOI: https://doi.org/10.1124/mol.57.3.512
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    Calcium-Independent Receptor for α-Latrotoxin and Neurexin 1α Facilitate Toxin-Induced Channel Formation: Evidence That Channel Formation Results from Tethering of Toxin to Membrane
    Michael D. Hlubek, Edward L. Stuenkel, Valery G. Krasnoperov, Alexander G. Petrenko and Ronald W. Holz
    Molecular Pharmacology March 2000, 57 (3) 519-528; DOI: https://doi.org/10.1124/mol.57.3.519
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    Effect of 6-Aminonicotinamide and Other Protein Synthesis Inhibitors on Formation of Platinum-DNA Adducts and Cisplatin Sensitivity
    I. Imawati Budihardjo, Scott A. Boerner, Steven Eckdahl, Phyllis A. Svingen, Robert Rios, Matthew M. Ames and Scott H. Kaufmann
    Molecular Pharmacology March 2000, 57 (3) 529-538; DOI: https://doi.org/10.1124/mol.57.3.529
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    Identification of Threonine Residues Controlling the Agonist-Dependent Phosphorylation and Desensitization of the Rat A3 Adenosine Receptor
    Timothy M. Palmer and Gary L. Stiles
    Molecular Pharmacology March 2000, 57 (3) 539-545; DOI: https://doi.org/10.1124/mol.57.3.539
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    Subtype-Specific Kinetics of Inhibitory Adenosine Receptor Internalization Are Determined by Sensitivity to Phosphorylation by G Protein-Coupled Receptor Kinases
    Gail Ferguson, Kenneth R. Watterson and Timothy M. Palmer
    Molecular Pharmacology March 2000, 57 (3) 546-552; DOI: https://doi.org/10.1124/mol.57.3.546
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    RPR112378 and RPR115781: Two Representatives of a New Family of Microtubule Assembly Inhibitors
    Cécile Combeau, Jean Provost, Frédérique Lancelin, Yann Tournoux, François Prod'homme, Frédéric Herman, François Lavelle, Jean Leboul and Marc Vuilhorgne
    Molecular Pharmacology March 2000, 57 (3) 553-563; DOI: https://doi.org/10.1124/mol.57.3.553
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    Calmodulin Increases the Sensitivity of Type 3 Inositol-1,4,5-trisphosphate Receptors to Ca2+ Inhibition in Human Bronchial Mucosal Cells
    Ludwig Missiaen, Humbert DeSmedt, Geert Bultynck, Sara Vanlingen, Patrick Desmet, Geert Callewaert and Jan B. Parys
    Molecular Pharmacology March 2000, 57 (3) 564-567; DOI: https://doi.org/10.1124/mol.57.3.564
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    A Steroid Derivative with Paclitaxel-Like Effects on Tubulin Polymerization
    Pascal Verdier-Pinard, Zhiqiang Wang, Arasambattu K. Mohanakrishnan, Mark Cushman and Ernest Hamel
    Molecular Pharmacology March 2000, 57 (3) 568-575; DOI: https://doi.org/10.1124/mol.57.3.568
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    Cloned Human Aquaporin-1 Is a Cyclic GMP-Gated Ion Channel
    Todd L. Anthony, Heddwen L. Brooks, Daniela Boassa, Sergey Leonov, Gina M. Yanochko, John W. Regan and Andrea J. Yool
    Molecular Pharmacology March 2000, 57 (3) 576-588; DOI: https://doi.org/10.1124/mol.57.3.576
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    Catechol-O-methyltransferase Inhibition Attenuates Levodopa Toxicity in Mesencephalic Dopamine Neurons
    Alexander Storch, Heike Blessing, Markus Bareiss, Sinje Jankowski, Zao Dung Ling, Paul Carvey and Johannes Schwarz
    Molecular Pharmacology March 2000, 57 (3) 589-594; DOI: https://doi.org/10.1124/mol.57.3.589
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    myo-Inositol 1,4,6-Trisphosphorothioate andmyo-Inositol 1,3,6-Trisphosphorothioate: Partial Agonists with Very Low Intrinsic Activity at the Plateletmyo-Inositol 1,4,5-Trisphosphate Receptor
    Christine T. Murphy, Andrew M. Riley, Steve J. Mills, Catherine J. Lindley, Barry V. L. Potter and John Westwick
    Molecular Pharmacology March 2000, 57 (3) 595-601; DOI: https://doi.org/10.1124/mol.57.3.595
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    Potency of Ligands Correlates with Affinity Measured against Agonist and Inverse Agonists but Not against Neutral Ligand in Constitutively Active Chemokine Receptor
    Mette M. Rosenkilde and Thue W. Schwartz
    Molecular Pharmacology March 2000, 57 (3) 602-609; DOI: https://doi.org/10.1124/mol.57.3.602
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    Transcriptional Induction of Heme Oxygenase-1 Gene Expression by Okadaic Acid in Primary Rat Hepatocyte Cultures
    Stephan Immenschuh, Vera Hinke, Norbert Katz and Thomas Kietzmann
    Molecular Pharmacology March 2000, 57 (3) 610-618; DOI: https://doi.org/10.1124/mol.57.3.610
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    The Human Glutathione Transferase P1-1 Specific Inhibitor TER 117 Designed for Overcoming Cytostatic-Drug Resistance Is also a Strong Inhibitor of Glyoxalase I
    Ann-Sofie Johansson, Marianne Ridderström and Bengt Mannervik
    Molecular Pharmacology March 2000, 57 (3) 619-624; DOI: https://doi.org/10.1124/mol.57.3.619
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    Functional Importance of Transmembrane Helix 6 Trp279and Exoloop 3 Val299 of Rat Gonadotropin-Releasing Hormone Receptor
    Stéphanie Chauvin, Annette Bérault, Yannick Lerrant, Marcel Hibert and Raymond Counis
    Molecular Pharmacology March 2000, 57 (3) 625-633; DOI: https://doi.org/10.1124/mol.57.3.625
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    Transport Function and Hepatocellular Localization of mrp6 in Rat Liver
    Jerzy Madon, Bruno Hagenbuch, Lukas Landmann, Peter J. Meier and Bruno Stieger
    Molecular Pharmacology March 2000, 57 (3) 634-641; DOI: https://doi.org/10.1124/mol.57.3.634

Accelerated Communication

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    5-Iodo-A-85380, an α4β2 Subtype-Selective Ligand for Nicotinic Acetylcholine Receptors
    Alexey G. Mukhin, Daniela Gündisch, Andrew G. Horti, Andrei O. Koren, Gilles Tamagnan, Alane S. Kimes, Joann Chambers, D. Bruce Vaupel, Sarah L. King, Marina R. Picciotto, Robert B. Innis and Edythe D. London
    Molecular Pharmacology March 2000, 57 (3) 642-649; DOI: https://doi.org/10.1124/mol.57.3.642
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Molecular Pharmacology: 57 (3)
Molecular Pharmacology
Vol. 57, Issue 3
1 Mar 2000
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