Table of Contents

Articles

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  Ca²⁺ Requirement for High-Affinity γ-Aminobutyric Acid (GABA) Binding at GABA_B Receptors: Involvement of Serine 269 of the GABA_BR1 Subunit

  Thierry Galvez, Stephan Urwyler, Laurent Prézeau, Johannes Mosbacher, Cécile Joly, Barbara Malitschek, Jakob Heid, Isabelle Brabet, Wolfgang Froestl, Bernhard Bettler, Klemens Kaupmann and Jean-Philippe Pin

  Molecular Pharmacology March 2000, 57 (3) 419-426; DOI: https://doi.org/10.1124/mol.57.3.419
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  Structure-Activity Relationship of Staurosporine Analogs in Regulating Expression of Endothelial Nitric-Oxide Synthase Gene

  Huige Li and Ulrich Förstermann

  Molecular Pharmacology March 2000, 57 (3) 427-435; DOI: https://doi.org/10.1124/mol.57.3.427
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  Allosteric Interactions between the Antagonist Prazosin and Amiloride Analogs at the Human α_1A-Adrenergic Receptor

  Ray A. Leppik, Anita Mynett, Sebastian Lazareno and Nigel J. M. Birdsall

  Molecular Pharmacology March 2000, 57 (3) 436-445; DOI: https://doi.org/10.1124/mol.57.3.436
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  Modulation of Dopamine D₂ Receptor Signaling by Actin-Binding Protein (ABP-280)

  M. Li, J. C. Bermak, Z. W. Wang and Q. Y. Zhou

  Molecular Pharmacology March 2000, 57 (3) 446-452; DOI: https://doi.org/10.1124/mol.57.3.446
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  Characterization of Protein Kinase chk1 Essential for the Cell Cycle Checkpoint after Exposure of Human Head and Neck Carcinoma A253 Cells to a Novel Topoisomerase I Inhibitor BNP1350

  Ming-Biao Yin, Bin Guo, Udo Vanhoefer, Rami G. Azrak, Hans Minderman, Cheryl Frank, Carol Wrzosek, Harry K. Slocum and Youcef M. Rustum

  Molecular Pharmacology March 2000, 57 (3) 453-459; DOI: https://doi.org/10.1124/mol.57.3.453
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  Specific Regulation of RGS2 Messenger RNA by Angiotensin II in Cultured Vascular Smooth Muscle Cells

  Sharon L. Grant, Bernard Lassègue, Kathy K. Griendling, Masuko Ushio-Fukai, P. Reid Lyons and R. Wayne Alexander

  Molecular Pharmacology March 2000, 57 (3) 460-467; DOI: https://doi.org/10.1124/mol.57.3.460
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  Substrate-Dependent Regulation of Human ArylamineN-Acetyltransferase-1 in Cultured Cells

  Neville J. Butcher, Kenneth F. Ilett and Rodney F. Minchin

  Molecular Pharmacology March 2000, 57 (3) 468-473; DOI: https://doi.org/10.1124/mol.57.3.468
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  A Single Glycine Residue at the Entrance to the First Membrane-Spanning Domain of the γ-Aminobutyric Acid Type A Receptor β₂ Subunit Affects Allosteric Sensitivity to GABA and Anesthetics

  Berit X. Carlson, A. Christine Engblom, Uffe Kristiansen, Arne Schousboe and Richard W. Olsen

  Molecular Pharmacology March 2000, 57 (3) 474-484; DOI: https://doi.org/10.1124/mol.57.3.474
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  Inhibition of c-myc Expression in Cells by Targeting an RNA-Protein Interaction Using Antisense Oligonucleotides

  Christopher M. Coulis, Chunja Lee, Violet Nardone and Rebecca D. Prokipcak

  Molecular Pharmacology March 2000, 57 (3) 485-494; DOI: https://doi.org/10.1124/mol.57.3.485
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  Functional Inactivation of the Nociceptin Receptor by Alanine Substitution of Glutamine 286 at the C Terminus of Transmembrane Segment VI: Evidence from a Site-Directed Mutagenesis Study of the ORL1 Receptor Transmembrane-Binding Domain

  Lionel Mouledous, Christopher M. Topham, Christiane Moisand, Catherine Mollereau and Jean-Claude Meunier

  Molecular Pharmacology March 2000, 57 (3) 495-502; DOI: https://doi.org/10.1124/mol.57.3.495
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  Effect of p53 Status on Sensitivity to Platinum Complexes in a Human Ovarian Cancer Cell Line

  Katharine E. Pestell, Stephen M. Hobbs, Jenny C. Titley, Lloyd R. Kelland and Michael I. Walton

  Molecular Pharmacology March 2000, 57 (3) 503-511; DOI: https://doi.org/10.1124/mol.57.3.503
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  Hematotoxicity of the Chinese Herbal Medicine Tripterygium wilfordii Hook f in CD34-Positive Human Bone Marrow Cells

  David W. Pyatt, Yanzhu Yang, Brenda Mehos, Anh Le, Wayne Stillman and Richard D. Irons

  Molecular Pharmacology March 2000, 57 (3) 512-518; DOI: https://doi.org/10.1124/mol.57.3.512
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  Calcium-Independent Receptor for α-Latrotoxin and Neurexin 1α Facilitate Toxin-Induced Channel Formation: Evidence That Channel Formation Results from Tethering of Toxin to Membrane

  Michael D. Hlubek, Edward L. Stuenkel, Valery G. Krasnoperov, Alexander G. Petrenko and Ronald W. Holz

  Molecular Pharmacology March 2000, 57 (3) 519-528; DOI: https://doi.org/10.1124/mol.57.3.519
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  Effect of 6-Aminonicotinamide and Other Protein Synthesis Inhibitors on Formation of Platinum-DNA Adducts and Cisplatin Sensitivity

  I. Imawati Budihardjo, Scott A. Boerner, Steven Eckdahl, Phyllis A. Svingen, Robert Rios, Matthew M. Ames and Scott H. Kaufmann

  Molecular Pharmacology March 2000, 57 (3) 529-538; DOI: https://doi.org/10.1124/mol.57.3.529
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  Identification of Threonine Residues Controlling the Agonist-Dependent Phosphorylation and Desensitization of the Rat A₃ Adenosine Receptor

  Timothy M. Palmer and Gary L. Stiles

  Molecular Pharmacology March 2000, 57 (3) 539-545; DOI: https://doi.org/10.1124/mol.57.3.539
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  Subtype-Specific Kinetics of Inhibitory Adenosine Receptor Internalization Are Determined by Sensitivity to Phosphorylation by G Protein-Coupled Receptor Kinases

  Gail Ferguson, Kenneth R. Watterson and Timothy M. Palmer

  Molecular Pharmacology March 2000, 57 (3) 546-552; DOI: https://doi.org/10.1124/mol.57.3.546
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  RPR112378 and RPR115781: Two Representatives of a New Family of Microtubule Assembly Inhibitors

  Cécile Combeau, Jean Provost, Frédérique Lancelin, Yann Tournoux, François Prod'homme, Frédéric Herman, François Lavelle, Jean Leboul and Marc Vuilhorgne

  Molecular Pharmacology March 2000, 57 (3) 553-563; DOI: https://doi.org/10.1124/mol.57.3.553
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  Calmodulin Increases the Sensitivity of Type 3 Inositol-1,4,5-trisphosphate Receptors to Ca²⁺ Inhibition in Human Bronchial Mucosal Cells

  Ludwig Missiaen, Humbert DeSmedt, Geert Bultynck, Sara Vanlingen, Patrick Desmet, Geert Callewaert and Jan B. Parys

  Molecular Pharmacology March 2000, 57 (3) 564-567; DOI: https://doi.org/10.1124/mol.57.3.564
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  A Steroid Derivative with Paclitaxel-Like Effects on Tubulin Polymerization

  Pascal Verdier-Pinard, Zhiqiang Wang, Arasambattu K. Mohanakrishnan, Mark Cushman and Ernest Hamel

  Molecular Pharmacology March 2000, 57 (3) 568-575; DOI: https://doi.org/10.1124/mol.57.3.568
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  Cloned Human Aquaporin-1 Is a Cyclic GMP-Gated Ion Channel

  Todd L. Anthony, Heddwen L. Brooks, Daniela Boassa, Sergey Leonov, Gina M. Yanochko, John W. Regan and Andrea J. Yool

  Molecular Pharmacology March 2000, 57 (3) 576-588; DOI: https://doi.org/10.1124/mol.57.3.576
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  Catechol-O-methyltransferase Inhibition Attenuates Levodopa Toxicity in Mesencephalic Dopamine Neurons

  Alexander Storch, Heike Blessing, Markus Bareiss, Sinje Jankowski, Zao Dung Ling, Paul Carvey and Johannes Schwarz

  Molecular Pharmacology March 2000, 57 (3) 589-594; DOI: https://doi.org/10.1124/mol.57.3.589
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  myo-Inositol 1,4,6-Trisphosphorothioate andmyo-Inositol 1,3,6-Trisphosphorothioate: Partial Agonists with Very Low Intrinsic Activity at the Plateletmyo-Inositol 1,4,5-Trisphosphate Receptor

  Christine T. Murphy, Andrew M. Riley, Steve J. Mills, Catherine J. Lindley, Barry V. L. Potter and John Westwick

  Molecular Pharmacology March 2000, 57 (3) 595-601; DOI: https://doi.org/10.1124/mol.57.3.595
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  Potency of Ligands Correlates with Affinity Measured against Agonist and Inverse Agonists but Not against Neutral Ligand in Constitutively Active Chemokine Receptor

  Mette M. Rosenkilde and Thue W. Schwartz

  Molecular Pharmacology March 2000, 57 (3) 602-609; DOI: https://doi.org/10.1124/mol.57.3.602
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  Transcriptional Induction of Heme Oxygenase-1 Gene Expression by Okadaic Acid in Primary Rat Hepatocyte Cultures

  Stephan Immenschuh, Vera Hinke, Norbert Katz and Thomas Kietzmann

  Molecular Pharmacology March 2000, 57 (3) 610-618; DOI: https://doi.org/10.1124/mol.57.3.610
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  The Human Glutathione Transferase P1-1 Specific Inhibitor TER 117 Designed for Overcoming Cytostatic-Drug Resistance Is also a Strong Inhibitor of Glyoxalase I

  Ann-Sofie Johansson, Marianne Ridderström and Bengt Mannervik

  Molecular Pharmacology March 2000, 57 (3) 619-624; DOI: https://doi.org/10.1124/mol.57.3.619
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  Functional Importance of Transmembrane Helix 6 Trp²⁷⁹and Exoloop 3 Val²⁹⁹ of Rat Gonadotropin-Releasing Hormone Receptor

  Stéphanie Chauvin, Annette Bérault, Yannick Lerrant, Marcel Hibert and Raymond Counis

  Molecular Pharmacology March 2000, 57 (3) 625-633; DOI: https://doi.org/10.1124/mol.57.3.625
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  Transport Function and Hepatocellular Localization of mrp6 in Rat Liver

  Jerzy Madon, Bruno Hagenbuch, Lukas Landmann, Peter J. Meier and Bruno Stieger

  Molecular Pharmacology March 2000, 57 (3) 634-641; DOI: https://doi.org/10.1124/mol.57.3.634