Table of Contents

June 2009; 75 (6)

MINIREVIEWS

    • Jamie L. McConnell and
    • Brian E. Wadzinski

    Targeting Protein Serine/Threonine Phosphatases for Drug Development

    Mol Pharmacol June 2009 75:1249-1261; published ahead of print March 19, 2009, doi:10.1124/mol.108.053140
    • Joris Vriens,
    • Giovanni Appendino,
    • and Bernd Nilius

    Pharmacology of Vanilloid Transient Receptor Potential Cation Channels

    Mol Pharmacol June 2009 75:1262-1279; published ahead of print March 18, 2009, doi:10.1124/mol.109.055624

Accelerated Communication

    • Masahiro Tsuda,
    • Tomohiro Terada,
    • Tomoyuki Mizuno,
    • Toshiya Katsura,
    • Jin Shimakura,
    • and Ken-ichi Inui

    Targeted Disruption of the Multidrug and Toxin Extrusion 1 (Mate1) Gene in Mice Reduces Renal Secretion of Metformin

    Mol Pharmacol June 2009 75:1280-1286; published ahead of print March 30, 2009, doi:10.1124/mol.109.056242

Articles

    • Kazuharu Furutani,
    • Yukihiro Ohno,
    • Atsushi Inanobe,
    • Hiroshi Hibino,
    • and Yoshihisa Kurachi

    Mutational and In Silico Analyses for Antidepressant Block of Astroglial Inward-Rectifier Kir4.1 Channel

    Mol Pharmacol June 2009 75:1287-1295; published ahead of print March 5, 2009, doi:10.1124/mol.108.052936
    • Jacqueline M. Fonseca and
    • Nevin A. Lambert

    Instability of a Class A G Protein-Coupled Receptor Oligomer Interface

    Mol Pharmacol June 2009 75:1296-1299; published ahead of print March 9, 2009, doi:10.1124/mol.108.053876
    • Jean-Marc Navenot,
    • Nobutaka Fujii,
    • and Stephen C. Peiper

    Activation of Rho and Rho-Associated Kinase by GPR54 and KiSS1 Metastasis Suppressor Gene Product Induces Changes of Cell Morphology and Contributes to Apoptosis

    Mol Pharmacol June 2009 75:1300-1306; published ahead of print March 13, 2009, doi:10.1124/mol.109.055095
    • Xin Ge,
    • Horace H. Loh,
    • and Ping-Yee Law

    μ-Opioid Receptor Cell Surface Expression Is Regulated by Its Direct Interaction with Ribophorin I

    Mol Pharmacol June 2009 75:1307-1316; published ahead of print March 16, 2009, doi:10.1124/mol.108.054064
    • Isabelle Petit-Topin,
    • Nathalie Turque,
    • Jérôme Fagart,
    • Michel Fay,
    • André Ulmann,
    • Erin Gainer,
    • and Marie-Edith Rafestin-Oblin

    Met909 Plays a Key Role in the Activation of the Progesterone Receptor and Also in the High Potency of 13-Ethyl Progestins

    Mol Pharmacol June 2009 75:1317-1324; published ahead of print March 16, 2009, doi:10.1124/mol.108.054312
    • Spencer E. Hall,
    • Allen Mao,
    • Vicky Nicolaidou,
    • Mattea Finelli,
    • Emma L. Wise,
    • Belinda Nedjai,
    • Julie Kanjanapangka,
    • Paymann Harirchian,
    • Deborah Chen,
    • Victor Selchau,
    • Sofia Ribeiro,
    • Sabine Schyler,
    • James E. Pease,
    • Richard Horuk,
    • and Nagarajan Vaidehi

    Elucidation of Binding Sites of Dual Antagonists in the Human Chemokine Receptors CCR2 and CCR5

    Mol Pharmacol June 2009 75:1325-1336; published ahead of print March 18, 2009, doi:10.1124/mol.108.053470
    • Matthew G. McDonald,
    • Mark J. Rieder,
    • Mariko Nakano,
    • Clara K. Hsia,
    • and Allan E. Rettie

    CYP4F2 Is a Vitamin K1 Oxidase: An Explanation for Altered Warfarin Dose in Carriers of the V433M Variant

    Mol Pharmacol June 2009 75:1337-1346; published ahead of print March 18, 2009, doi:10.1124/mol.109.054833
    • Samantha McCavera,
    • Adrian T. Rogers,
    • Darran M. Yates,
    • Debra J. Woods,
    • and Adrian J. Wolstenholme

    An Ivermectin-Sensitive Glutamate-Gated Chloride Channel from the Parasitic Nematode Haemonchus contortus

    Mol Pharmacol June 2009 75:1347-1355; published ahead of print March 31, 2009, doi:10.1124/mol.108.053363
    • B. Cui,
    • S. P. Johnson,
    • N. Bullock,
    • F. Ali-Osman,
    • D. D. Bigner,
    • and H. S. Friedman

    Bifunctional DNA Alkylator 1,3-Bis(2-chloroethyl)-1-nitrosourea Activates the ATR-Chk1 Pathway Independently of the Mismatch Repair Pathway

    Mol Pharmacol June 2009 75:1356-1363; published ahead of print March 4, 2009, doi:10.1124/mol.108.053124
    • Le Yu,
    • William Ka Kei Wu,
    • Zhi Jie Li,
    • Qi Cai Liu,
    • Hai Tao Li,
    • Ya Chun Wu,
    • and Chi Hin Cho

    Enhancement of Doxorubicin Cytotoxicity on Human Esophageal Squamous Cell Carcinoma Cells by Indomethacin and 4-[5-(4-Chlorophenyl)-3-(trifluoromethyl)-1H-pyrazol-1-yl]benzenesulfonamide (SC236) via Inhibiting P-Glycoprotein Activity

    Mol Pharmacol June 2009 75:1364-1373; published ahead of print March 5, 2009, doi:10.1124/mol.108.053546
    • Yu-Zhuo Pan,
    • Marilyn E. Morris,
    • and Ai-Ming Yu

    MicroRNA-328 Negatively Regulates the Expression of Breast Cancer Resistance Protein (BCRP/ABCG2) in Human Cancer Cells

    Mol Pharmacol June 2009 75:1374-1379; published ahead of print March 6, 2009, doi:10.1124/mol.108.054163
    • José Brea,
    • Marián Castro,
    • Jesús Giraldo,
    • Juan F. López-Giménez,
    • Juan Fernando Padín,
    • Fátima Quintián,
    • Maria Isabel Cadavid,
    • Maria Teresa Vilaró,
    • Guadalupe Mengod,
    • Kelly A. Berg,
    • William P. Clarke,
    • Jean-Pierre Vilardaga,
    • Graeme Milligan,
    • and Maria Isabel Loza

    Evidence for Distinct Antagonist-Revealed Functional States of 5-Hydroxytryptamine2A Receptor Homodimers

    Mol Pharmacol June 2009 75:1380-1391; published ahead of print March 11, 2009, doi:10.1124/mol.108.054395
    • Maria Ellfolk,
    • Maria Norlin,
    • Katarina Gyllensten,
    • and Kjell Wikvall

    Regulation of Human Vitamin D3 25-Hydroxylases in Dermal Fibroblasts and Prostate Cancer LNCaP Cells

    Mol Pharmacol June 2009 75:1392-1399; published ahead of print March 13, 2009, doi:10.1124/mol.108.053660
    • Gustav Akk,
    • Ping Li,
    • John Bracamontes,
    • and Joe Henry Steinbach

    Activation and Modulation of Concatemeric GABA-A Receptors Expressed in Human Embryonic Kidney Cells

    Mol Pharmacol June 2009 75:1400-1411; published ahead of print March 16, 2009, doi:10.1124/mol.108.054510
    • Colin A. Flaveny,
    • Iain A. Murray,
    • Chris R. Chiaro,
    • and Gary H. Perdew

    Ligand Selectivity and Gene Regulation by the Human Aryl Hydrocarbon Receptor in Transgenic Mice

    Mol Pharmacol June 2009 75:1412-1420; published ahead of print March 19, 2009, doi:10.1124/mol.109.054825
    • Andrea Kromer and
    • Bernd Moosmann

    Statin-Induced Liver Injury Involves Cross-Talk between Cholesterol and Selenoprotein Biosynthetic Pathways

    Mol Pharmacol June 2009 75:1421-1429; published ahead of print March 30, 2009, doi:10.1124/mol.108.053678
    • Leigh Wellhauser,
    • Patrick Kim Chiaw,
    • Stan Pasyk,
    • Canhui Li,
    • Mohabir Ramjeesingh,
    • and Christine E. Bear

    A Small-Molecule Modulator Interacts Directly with ΔPhe508-CFTR to Modify Its ATPase Activity and Conformational Stability

    Mol Pharmacol June 2009 75:1430-1438; published ahead of print April 1, 2009, doi:10.1124/mol.109.055608

Cover image

Cover image expansion

About the cover: Effect of mutations at Gln150 and Leu151 on Kir4.1 channel currents and block. See the article by Furutani et al. on page 1287 of this issue.

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June 2009; 75 (6)
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