Table of Contents

July 2009; 76 (1)

MINIREVIEW

    • Kazuhiko Matsuda,
    • Satoshi Kanaoka,
    • Miki Akamatsu,
    • and David B. Sattelle

    Diverse Actions and Target-Site Selectivity of Neonicotinoids: Structural Insights

    Mol Pharmacol July 2009 76:1-10; published ahead of print March 25, 2009, doi:10.1124/mol.109.055186
    • Marla L. Yates and
    • Eric L. Barker

    Inactivation and Biotransformation of the Endogenous Cannabinoids Anandamide and 2-Arachidonoylglycerol

    Mol Pharmacol July 2009 76:11-17; published ahead of print April 23, 2009, doi:10.1124/mol.109.055251

Accelerated Communication

    • Laura K. K. Pacey,
    • Scott P. Heximer,
    • and David R. Hampson

    Increased GABAB Receptor-Mediated Signaling Reduces the Susceptibility of Fragile X Knockout Mice to Audiogenic Seizures

    Mol Pharmacol July 2009 76:18-24; published ahead of print April 7, 2009, doi:10.1124/mol.109.056127

Articles

    • Hans-Joachim Wittmann,
    • Roland Seifert,
    • and Andrea Strasser

    Contribution of Binding Enthalpy and Entropy to Affinity of Antagonist and Agonist Binding at Human and Guinea Pig Histamine H1-Receptor

    Mol Pharmacol July 2009 76:25-37; published ahead of print April 3, 2009, doi:10.1124/mol.109.055384
    • Seung-Kuy Cha,
    • Ming-Chang Hu,
    • Hiroshi Kurosu,
    • Makoto Kuro-o,
    • Orson Moe,
    • and Chou-Long Huang

    Regulation of Renal Outer Medullary Potassium Channel and Renal K+ Excretion by Klotho

    Mol Pharmacol July 2009 76:38-46; published ahead of print April 6, 2009, doi:10.1124/mol.109.055780
    • Shuo Wei,
    • Hsiao-Ching Chuang,
    • Wan-Chi Tsai,
    • Hsiao-Ching Yang,
    • Shiuh-Rong Ho,
    • Andrew J. Paterson,
    • Samuel K. Kulp,
    • and Ching-Shih Chen

    Thiazolidinediones Mimic Glucose Starvation in Facilitating Sp1 Degradation through the Up-Regulation of β-Transducin Repeat-Containing Protein

    Mol Pharmacol July 2009 76:47-57; published ahead of print April 16, 2009, doi:10.1124/mol.109.055376
    • Ester Gutiérrez-Pascual,
    • Jérôme Leprince,
    • Antonio J. Martínez-Fuentes,
    • Isabelle Ségalas-Milazzo,
    • Rafael Pineda,
    • Juan Roa,
    • Mario Duran-Prado,
    • Laure Guilhaudis,
    • Elia Desperrois,
    • Aurélie Lebreton,
    • Leonor Pinilla,
    • Marie-Christine Tonon,
    • María M. Malagón,
    • Hubert Vaudry,
    • Manuel Tena-Sempere,
    • and Justo P. Castaño

    In Vivo and in Vitro Structure-Activity Relationships and Structural Conformation of Kisspeptin-10-Related Peptides

    Mol Pharmacol July 2009 76:58-67; published ahead of print April 23, 2009, doi:10.1124/mol.108.053751
    • Qisheng Liu,
    • Mark S. Bee,
    • and Agnes Schonbrunn

    Site Specificity of Agonist and Second Messenger-Activated Kinases for Somatostatin Receptor Subtype 2A (Sst2A) Phosphorylation

    Mol Pharmacol July 2009 76:68-80; published ahead of print April 23, 2009, doi:10.1124/mol.108.054262
    • Jun Li,
    • Yun Wang,
    • Chaozhe Yang,
    • Pengfei Wang,
    • Denise K. Oelschlager,
    • Yong Zheng,
    • De-An Tian,
    • William E. Grizzle,
    • Donald J. Buchsbaum,
    • and Mei Wan

    Polyethylene Glycosylated Curcumin Conjugate Inhibits Pancreatic Cancer Cell Growth through Inactivation of Jab1

    Mol Pharmacol July 2009 76:81-90; published ahead of print April 24, 2009, doi:10.1124/mol.109.054551
    • Yanxia Liu,
    • Brian K. Law,
    • and Hendrik Luesch

    Apratoxin A Reversibly Inhibits the Secretory Pathway by Preventing Cotranslational Translocation

    Mol Pharmacol July 2009 76:91-104; published ahead of print April 29, 2009, doi:10.1124/mol.109.056085
    • Elton Migliati,
    • Nathalie Meurice,
    • Pascale DuBois,
    • Jennifer S. Fang,
    • Suma Somasekharan,
    • Elizabeth Beckett,
    • Gary Flynn,
    • and Andrea J. Yool

    Inhibition of Aquaporin-1 and Aquaporin-4 Water Permeability by a Derivative of the Loop Diuretic Bumetanide Acting at an Internal Pore-Occluding Binding Site

    Mol Pharmacol July 2009 76:105-112; published ahead of print April 29, 2009, doi:10.1124/mol.108.053744
    • Louise M. Hughes,
    • Renate Griffith,
    • Alison Carey,
    • Trent Butler,
    • Scott W. Donne,
    • Ken W. Beagley,
    • and R. John Aitken

    The Spermostatic and Microbicidal Actions of Quinones and Maleimides: Toward a Dual-Purpose Contraceptive Agent

    Mol Pharmacol July 2009 76:113-124; published ahead of print March 31, 2009, doi:10.1124/mol.108.053645
    • Christopher V. DeSimone,
    • YiChun Lu,
    • Vladimir E. Bondarenko,
    • and Michael J. Morales

    S3b Amino Acid Substitutions and Ancillary Subunits Alter the Affinity of Heteropoda venatoria Toxin 2 for Kv4.3

    Mol Pharmacol July 2009 76:125-133; published ahead of print April 8, 2009, doi:10.1124/mol.109.055657
    • Wendy Walwyn,
    • Scott John,
    • Matthew Maga,
    • Christopher J. Evans,
    • and Tim G. Hales

    δ Receptors Are Required for Full Inhibitory Coupling of μ Receptors to Voltage-Dependent Ca2+ Channels in Dorsal Root Ganglion Neurons

    Mol Pharmacol July 2009 76:134-143; published ahead of print April 8, 2009, doi:10.1124/mol.109.055913
    • Dianne M. Perez,
    • Robert S. Papay,
    • and Ting Shi

    α1-Adrenergic Receptor Stimulates Interleukin-6 Expression and Secretion through Both mRNA Stability and Transcriptional Regulation: Involvement of p38 Mitogen-Activated Protein Kinase and Nuclear Factor-κB

    Mol Pharmacol July 2009 76:144-152; published ahead of print April 10, 2009, doi:10.1124/mol.108.054320
    • Kent T. Symons,
    • Mark E. Massari,
    • Phan M. Nguyen,
    • Tom T. Lee,
    • Jeffrey Roppe,
    • Céline Bonnefous,
    • Joseph E. Payne,
    • Nicholas D. Smith,
    • Stewart A. Noble,
    • Marciano Sablad,
    • Natasha Rozenkrants,
    • Yan Zhang,
    • Tadimeti S. Rao,
    • Andrew K. Shiau,
    • and Christian A. Hassig

    KLYP956 Is a Non-Imidazole-Based Orally Active Inhibitor of Nitric-Oxide Synthase Dimerization

    Mol Pharmacol July 2009 76:153-162; published ahead of print April 13, 2009, doi:10.1124/mol.109.055434
    • Chao Yan,
    • Biehuoy Shieh,
    • Philip Reigan,
    • Zhiyong Zhang,
    • Marie A. Colucci,
    • Aurélie Chilloux,
    • Jeffery J. Newsome,
    • David Siegel,
    • Dan Chan,
    • Christopher J. Moody,
    • and David Ross

    Potent Activity of Indolequinones against Human Pancreatic Cancer: Identification of Thioredoxin Reductase as a Potential Target

    Mol Pharmacol July 2009 76:163-172; published ahead of print April 13, 2009, doi:10.1124/mol.109.055855
    • Konstantin Tsoyi,
    • Tae Yu Lee,
    • Young Soo Lee,
    • Hye Jung Kim,
    • Han Geuk Seo,
    • Jae Heun Lee,
    • and Ki Churl Chang

    Heme-Oxygenase-1 Induction and Carbon Monoxide-Releasing Molecule Inhibit Lipopolysaccharide (LPS)-Induced High-Mobility Group Box 1 Release in Vitro and Improve Survival of Mice in LPS- and Cecal Ligation and Puncture-Induced Sepsis Model in Vivo

    Mol Pharmacol July 2009 76:173-182; published ahead of print April 14, 2009, doi:10.1124/mol.109.055137
    • Koushik K. Das,
    • Manisha Bajpai,
    • Yingxin Kong,
    • Jianying Liu,
    • Xin Geng,
    • and Kiron M. Das

    Mesalamine Suppresses the Expression of TC22, a Novel Tropomyosin Isoform Associated with Colonic Neoplasia

    Mol Pharmacol July 2009 76:183-191; published ahead of print April 15, 2009, doi:10.1124/mol.109.056028
    • Tony W. H. Li,
    • Qingsong Zhang,
    • Pilsoo Oh,
    • Meng Xia,
    • Hui Chen,
    • Sean Bemanian,
    • Natalie Lastra,
    • Magda Circ,
    • Mary Pat Moyer,
    • José M. Mato,
    • Tak Yee Aw,
    • and Shelly C. Lu

    S-Adenosylmethionine and Methylthioadenosine Inhibit Cellular FLICE Inhibitory Protein Expression and Induce Apoptosis in Colon Cancer Cells

    Mol Pharmacol July 2009 76:192-200; published ahead of print April 16, 2009, doi:10.1124/mol.108.054411
    • Masataka Yanagawa,
    • Takahiro Yamashita,
    • and Yoshinori Shichida

    Activation Switch in the Transmembrane Domain of Metabotropic Glutamate Receptor

    Mol Pharmacol July 2009 76:201-207; published ahead of print April 27, 2009, doi:10.1124/mol.109.056549
    • Jill M. Wagner and
    • Larry M. Karnitz

    Cisplatin-Induced DNA Damage Activates Replication Checkpoint Signaling Components that Differentially Affect Tumor Cell Survival

    Mol Pharmacol July 2009 76:208-214; published ahead of print April 29, 2009, doi:10.1124/mol.109.055178

Cover image

Cover image expansion

About the cover: Electrostatic (A and B) and hydrogen bonding (C and D) fields extended from the ligand binding site of the peach potato aphid M. persicae (A and C) and the honeybee A. mellifera (B and D). See the article by Matsuda et al. on page 1 of this issue.

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July 2009; 76 (1)
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