Research ArticleArticle
Discovery and Mapping of an Intracellular Antagonist Binding Site at the Chemokine Receptor CCR2
Annelien J.M. Zweemer, Julia Bunnik, Margo Veenhuizen, Fabiana Miraglia, Eelke B. Lenselink, Maris Vilums, Henk de Vries, Arthur Gibert, Stefanie Thiele, Mette M. Rosenkilde, Adriaan P. IJzerman and Laura H. Heitman
Molecular Pharmacology October 2014, 86 (4) 358-368; DOI: https://doi.org/10.1124/mol.114.093328
Annelien J.M. Zweemer
Division of Medicinal Chemistry, Leiden Academic Centre for Drug Research, Leiden University, Leiden, the Netherlands (A.J.M.Z., J.B., M.V., F.M., E.B.L., M.V., H.V., A.G., A.P.IJ., L.H.H.); Laboratory for Molecular Pharmacology, Department of Neuroscience and Pharmacology, Faculty of Health and Medical Sciences, University of Copenhagen, Copenhagen, Denmark (S.T., M.M.R.)
Julia Bunnik
Division of Medicinal Chemistry, Leiden Academic Centre for Drug Research, Leiden University, Leiden, the Netherlands (A.J.M.Z., J.B., M.V., F.M., E.B.L., M.V., H.V., A.G., A.P.IJ., L.H.H.); Laboratory for Molecular Pharmacology, Department of Neuroscience and Pharmacology, Faculty of Health and Medical Sciences, University of Copenhagen, Copenhagen, Denmark (S.T., M.M.R.)
Margo Veenhuizen
Division of Medicinal Chemistry, Leiden Academic Centre for Drug Research, Leiden University, Leiden, the Netherlands (A.J.M.Z., J.B., M.V., F.M., E.B.L., M.V., H.V., A.G., A.P.IJ., L.H.H.); Laboratory for Molecular Pharmacology, Department of Neuroscience and Pharmacology, Faculty of Health and Medical Sciences, University of Copenhagen, Copenhagen, Denmark (S.T., M.M.R.)
Fabiana Miraglia
Division of Medicinal Chemistry, Leiden Academic Centre for Drug Research, Leiden University, Leiden, the Netherlands (A.J.M.Z., J.B., M.V., F.M., E.B.L., M.V., H.V., A.G., A.P.IJ., L.H.H.); Laboratory for Molecular Pharmacology, Department of Neuroscience and Pharmacology, Faculty of Health and Medical Sciences, University of Copenhagen, Copenhagen, Denmark (S.T., M.M.R.)
Eelke B. Lenselink
Division of Medicinal Chemistry, Leiden Academic Centre for Drug Research, Leiden University, Leiden, the Netherlands (A.J.M.Z., J.B., M.V., F.M., E.B.L., M.V., H.V., A.G., A.P.IJ., L.H.H.); Laboratory for Molecular Pharmacology, Department of Neuroscience and Pharmacology, Faculty of Health and Medical Sciences, University of Copenhagen, Copenhagen, Denmark (S.T., M.M.R.)
Maris Vilums
Division of Medicinal Chemistry, Leiden Academic Centre for Drug Research, Leiden University, Leiden, the Netherlands (A.J.M.Z., J.B., M.V., F.M., E.B.L., M.V., H.V., A.G., A.P.IJ., L.H.H.); Laboratory for Molecular Pharmacology, Department of Neuroscience and Pharmacology, Faculty of Health and Medical Sciences, University of Copenhagen, Copenhagen, Denmark (S.T., M.M.R.)
Henk de Vries
Division of Medicinal Chemistry, Leiden Academic Centre for Drug Research, Leiden University, Leiden, the Netherlands (A.J.M.Z., J.B., M.V., F.M., E.B.L., M.V., H.V., A.G., A.P.IJ., L.H.H.); Laboratory for Molecular Pharmacology, Department of Neuroscience and Pharmacology, Faculty of Health and Medical Sciences, University of Copenhagen, Copenhagen, Denmark (S.T., M.M.R.)
Arthur Gibert
Division of Medicinal Chemistry, Leiden Academic Centre for Drug Research, Leiden University, Leiden, the Netherlands (A.J.M.Z., J.B., M.V., F.M., E.B.L., M.V., H.V., A.G., A.P.IJ., L.H.H.); Laboratory for Molecular Pharmacology, Department of Neuroscience and Pharmacology, Faculty of Health and Medical Sciences, University of Copenhagen, Copenhagen, Denmark (S.T., M.M.R.)
Stefanie Thiele
Division of Medicinal Chemistry, Leiden Academic Centre for Drug Research, Leiden University, Leiden, the Netherlands (A.J.M.Z., J.B., M.V., F.M., E.B.L., M.V., H.V., A.G., A.P.IJ., L.H.H.); Laboratory for Molecular Pharmacology, Department of Neuroscience and Pharmacology, Faculty of Health and Medical Sciences, University of Copenhagen, Copenhagen, Denmark (S.T., M.M.R.)
Mette M. Rosenkilde
Division of Medicinal Chemistry, Leiden Academic Centre for Drug Research, Leiden University, Leiden, the Netherlands (A.J.M.Z., J.B., M.V., F.M., E.B.L., M.V., H.V., A.G., A.P.IJ., L.H.H.); Laboratory for Molecular Pharmacology, Department of Neuroscience and Pharmacology, Faculty of Health and Medical Sciences, University of Copenhagen, Copenhagen, Denmark (S.T., M.M.R.)
Adriaan P. IJzerman
Division of Medicinal Chemistry, Leiden Academic Centre for Drug Research, Leiden University, Leiden, the Netherlands (A.J.M.Z., J.B., M.V., F.M., E.B.L., M.V., H.V., A.G., A.P.IJ., L.H.H.); Laboratory for Molecular Pharmacology, Department of Neuroscience and Pharmacology, Faculty of Health and Medical Sciences, University of Copenhagen, Copenhagen, Denmark (S.T., M.M.R.)
Laura H. Heitman
Division of Medicinal Chemistry, Leiden Academic Centre for Drug Research, Leiden University, Leiden, the Netherlands (A.J.M.Z., J.B., M.V., F.M., E.B.L., M.V., H.V., A.G., A.P.IJ., L.H.H.); Laboratory for Molecular Pharmacology, Department of Neuroscience and Pharmacology, Faculty of Health and Medical Sciences, University of Copenhagen, Copenhagen, Denmark (S.T., M.M.R.)
Submit a Response to This Article
Jump to comment:
No eLetters have been published for this article.
In this issue
Research ArticleArticle
Intracellular Binding Site at the Chemokine Receptor CCR2
Annelien J.M. Zweemer, Julia Bunnik, Margo Veenhuizen, Fabiana Miraglia, Eelke B. Lenselink, Maris Vilums, Henk de Vries, Arthur Gibert, Stefanie Thiele, Mette M. Rosenkilde, Adriaan P. IJzerman and Laura H. Heitman
Molecular Pharmacology October 1, 2014, 86 (4) 358-368; DOI: https://doi.org/10.1124/mol.114.093328
Research ArticleArticle
Intracellular Binding Site at the Chemokine Receptor CCR2
Annelien J.M. Zweemer, Julia Bunnik, Margo Veenhuizen, Fabiana Miraglia, Eelke B. Lenselink, Maris Vilums, Henk de Vries, Arthur Gibert, Stefanie Thiele, Mette M. Rosenkilde, Adriaan P. IJzerman and Laura H. Heitman
Molecular Pharmacology October 1, 2014, 86 (4) 358-368; DOI: https://doi.org/10.1124/mol.114.093328
Jump to section
Related Articles
Cited By...
More in this TOC Section
Similar Articles
Advertisement