Research ArticleArticle
Leflunomide Increases Hepatic Exposure to Methotrexate and Its Metabolite by Differentially Regulating Multidrug Resistance–Associated Protein Mrp2/3/4 Transporters via Peroxisome Proliferator–Activated Receptor α Activation
Le Wang, Leilei Ma, Yunfei Lin, Xing Liu, Ling Xiao, Yiting Zhang, Ye Xu, Hu Zhou and Guoyu Pan
Molecular Pharmacology June 2018, 93 (6) 563-574; DOI: https://doi.org/10.1124/mol.117.110593
Le Wang
Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai, China and University of Chinese Academy of Sciences, Beijing, China
Leilei Ma
Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai, China and University of Chinese Academy of Sciences, Beijing, China
Yunfei Lin
Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai, China and University of Chinese Academy of Sciences, Beijing, China
Xing Liu
Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai, China and University of Chinese Academy of Sciences, Beijing, China
Ling Xiao
Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai, China and University of Chinese Academy of Sciences, Beijing, China
Yiting Zhang
Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai, China and University of Chinese Academy of Sciences, Beijing, China
Ye Xu
Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai, China and University of Chinese Academy of Sciences, Beijing, China
Hu Zhou
Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai, China and University of Chinese Academy of Sciences, Beijing, China
Guoyu Pan
Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai, China and University of Chinese Academy of Sciences, Beijing, China
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Research ArticleArticle
Leflunomide Increases Methotrexate Exposure by Altering Mrps
Le Wang, Leilei Ma, Yunfei Lin, Xing Liu, Ling Xiao, Yiting Zhang, Ye Xu, Hu Zhou and Guoyu Pan
Molecular Pharmacology June 1, 2018, 93 (6) 563-574; DOI: https://doi.org/10.1124/mol.117.110593
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