Index by author
September 01, 2018; Volume 94,Issue 3
A
Alpsoy, Aktan
- You have accessA Novel CRISPR/Cas9-Based Cellular Model to Explore Adenylyl Cyclase and cAMP SignalingMonica Soto-Velasquez, Michael P. Hayes, Aktan Alpsoy, Emily C. Dykhuizen and Val J. WattsMolecular Pharmacology September 2018, 94 (3) 963-972; DOI: https://doi.org/10.1124/mol.118.111849
Altonsy, Mohammed O.
- You have accessLong-Acting β2-Adrenoceptor Agonists Enhance Glucocorticoid Receptor (GR)–Mediated Transcription by Gene-Specific Mechanisms Rather Than Generic Effects via GRChristopher F. Rider, Mohammed O. Altonsy, Mahmoud M. Mostafa, Suharsh V. Shah, Sarah Sasse, Martijn L. Manson, Dong Yan, Carina Kärrman-Mårdh, Anna Miller-Larsson, Anthony N. Gerber, Mark A. Giembycz and Robert NewtonMolecular Pharmacology September 2018, 94 (3) 1031-1046; DOI: https://doi.org/10.1124/mol.118.112755
Arama, May
- You have accessAn Outward-Facing Aromatic Amino Acid Is Crucial for Signaling between the Membrane-Spanning and Nucleotide-Binding Domains of Multidrug Resistance Protein 1 (MRP1; ABCC1)Kevin E. Weigl, Gwenaëlle Conseil, Alice J. Rothnie, May Arama, Yossi Tsfadia and Susan P. C. ColeMolecular Pharmacology September 2018, 94 (3) 1069-1078; DOI: https://doi.org/10.1124/mol.118.112615
B
Bdioui, Sara
- You have accessEquilibrium Assays Are Required to Accurately Characterize the Activity Profiles of Drugs Modulating Gq-Protein-Coupled ReceptorsSara Bdioui, Julien Verdi, Nicolas Pierre, Eric Trinquet, Thomas Roux and Terry KenakinMolecular Pharmacology September 2018, 94 (3) 992-1006; DOI: https://doi.org/10.1124/mol.118.112573
Beech, Alison J.
- You have accessSmall-Molecule G Protein–Coupled Receptor Kinase Inhibitors Attenuate G Protein–Coupled Receptor Kinase 2–Mediated Desensitization of Vasoconstrictor-Induced Arterial ContractionsRichard D. Rainbow, Sean Brennan, Robert Jackson, Alison J. Beech, Amal Bengreed, Helen V. Waldschmidt, John J. G. Tesmer, R. A. John Challiss and Jonathon M. WilletsMolecular Pharmacology September 2018, 94 (3) 1079-1091; DOI: https://doi.org/10.1124/mol.118.112524
Bengreed, Amal
- You have accessSmall-Molecule G Protein–Coupled Receptor Kinase Inhibitors Attenuate G Protein–Coupled Receptor Kinase 2–Mediated Desensitization of Vasoconstrictor-Induced Arterial ContractionsRichard D. Rainbow, Sean Brennan, Robert Jackson, Alison J. Beech, Amal Bengreed, Helen V. Waldschmidt, John J. G. Tesmer, R. A. John Challiss and Jonathon M. WilletsMolecular Pharmacology September 2018, 94 (3) 1079-1091; DOI: https://doi.org/10.1124/mol.118.112524
Bonaventure, Pascal
- Open AccessThe Zinc Transporter SLC39A7 (ZIP7) Is Essential for Regulation of Cytosolic Zinc LevelsGrace Woodruff, Christian G. Bouwkamp, Femke M. de Vrij, Timothy Lovenberg, Pascal Bonaventure, Steven A. Kushner and Anthony W. HarringtonMolecular Pharmacology September 2018, 94 (3) 1092-1100; DOI: https://doi.org/10.1124/mol.118.112557
Bouwkamp, Christian G.
- Open AccessThe Zinc Transporter SLC39A7 (ZIP7) Is Essential for Regulation of Cytosolic Zinc LevelsGrace Woodruff, Christian G. Bouwkamp, Femke M. de Vrij, Timothy Lovenberg, Pascal Bonaventure, Steven A. Kushner and Anthony W. HarringtonMolecular Pharmacology September 2018, 94 (3) 1092-1100; DOI: https://doi.org/10.1124/mol.118.112557
Brennan, Sean
- You have accessSmall-Molecule G Protein–Coupled Receptor Kinase Inhibitors Attenuate G Protein–Coupled Receptor Kinase 2–Mediated Desensitization of Vasoconstrictor-Induced Arterial ContractionsRichard D. Rainbow, Sean Brennan, Robert Jackson, Alison J. Beech, Amal Bengreed, Helen V. Waldschmidt, John J. G. Tesmer, R. A. John Challiss and Jonathon M. WilletsMolecular Pharmacology September 2018, 94 (3) 1079-1091; DOI: https://doi.org/10.1124/mol.118.112524
C
Challiss, R. A. John
- You have accessSmall-Molecule G Protein–Coupled Receptor Kinase Inhibitors Attenuate G Protein–Coupled Receptor Kinase 2–Mediated Desensitization of Vasoconstrictor-Induced Arterial ContractionsRichard D. Rainbow, Sean Brennan, Robert Jackson, Alison J. Beech, Amal Bengreed, Helen V. Waldschmidt, John J. G. Tesmer, R. A. John Challiss and Jonathon M. WilletsMolecular Pharmacology September 2018, 94 (3) 1079-1091; DOI: https://doi.org/10.1124/mol.118.112524
Chen, Jie
- Open AccessAllergen Delivery Inhibitors: A Rationale for Targeting Sentinel Innate Immune Signaling of Group 1 House Dust Mite Allergens through Structure-Based Protease Inhibitor DesignJihui Zhang, Jie Chen, Gary K. Newton, Trevor R. Perrior and Clive RobinsonMolecular Pharmacology September 2018, 94 (3) 1007-1030; DOI: https://doi.org/10.1124/mol.118.112730
Clark, Alex M.
- You have accessAssessment of Substrate-Dependent Ligand Interactions at the Organic Cation Transporter OCT2 Using Six Model SubstratesPhilip J. Sandoval, Kimberley M. Zorn, Alex M. Clark, Sean Ekins and Stephen H. WrightMolecular Pharmacology September 2018, 94 (3) 1057-1068; DOI: https://doi.org/10.1124/mol.117.111443
Cole, Susan P. C.
- You have accessAn Outward-Facing Aromatic Amino Acid Is Crucial for Signaling between the Membrane-Spanning and Nucleotide-Binding Domains of Multidrug Resistance Protein 1 (MRP1; ABCC1)Kevin E. Weigl, Gwenaëlle Conseil, Alice J. Rothnie, May Arama, Yossi Tsfadia and Susan P. C. ColeMolecular Pharmacology September 2018, 94 (3) 1069-1078; DOI: https://doi.org/10.1124/mol.118.112615
Conseil, Gwenaëlle
- You have accessAn Outward-Facing Aromatic Amino Acid Is Crucial for Signaling between the Membrane-Spanning and Nucleotide-Binding Domains of Multidrug Resistance Protein 1 (MRP1; ABCC1)Kevin E. Weigl, Gwenaëlle Conseil, Alice J. Rothnie, May Arama, Yossi Tsfadia and Susan P. C. ColeMolecular Pharmacology September 2018, 94 (3) 1069-1078; DOI: https://doi.org/10.1124/mol.118.112615
D
de Vrij, Femke M.
- Open AccessThe Zinc Transporter SLC39A7 (ZIP7) Is Essential for Regulation of Cytosolic Zinc LevelsGrace Woodruff, Christian G. Bouwkamp, Femke M. de Vrij, Timothy Lovenberg, Pascal Bonaventure, Steven A. Kushner and Anthony W. HarringtonMolecular Pharmacology September 2018, 94 (3) 1092-1100; DOI: https://doi.org/10.1124/mol.118.112557
Dykhuizen, Emily C.
- You have accessA Novel CRISPR/Cas9-Based Cellular Model to Explore Adenylyl Cyclase and cAMP SignalingMonica Soto-Velasquez, Michael P. Hayes, Aktan Alpsoy, Emily C. Dykhuizen and Val J. WattsMolecular Pharmacology September 2018, 94 (3) 963-972; DOI: https://doi.org/10.1124/mol.118.111849
E
Ekins, Sean
- You have accessAssessment of Substrate-Dependent Ligand Interactions at the Organic Cation Transporter OCT2 Using Six Model SubstratesPhilip J. Sandoval, Kimberley M. Zorn, Alex M. Clark, Sean Ekins and Stephen H. WrightMolecular Pharmacology September 2018, 94 (3) 1057-1068; DOI: https://doi.org/10.1124/mol.117.111443
G
Gerber, Anthony N.
- You have accessLong-Acting β2-Adrenoceptor Agonists Enhance Glucocorticoid Receptor (GR)–Mediated Transcription by Gene-Specific Mechanisms Rather Than Generic Effects via GRChristopher F. Rider, Mohammed O. Altonsy, Mahmoud M. Mostafa, Suharsh V. Shah, Sarah Sasse, Martijn L. Manson, Dong Yan, Carina Kärrman-Mårdh, Anna Miller-Larsson, Anthony N. Gerber, Mark A. Giembycz and Robert NewtonMolecular Pharmacology September 2018, 94 (3) 1031-1046; DOI: https://doi.org/10.1124/mol.118.112755
Giembycz, Mark A.
- You have accessLong-Acting β2-Adrenoceptor Agonists Enhance Glucocorticoid Receptor (GR)–Mediated Transcription by Gene-Specific Mechanisms Rather Than Generic Effects via GRChristopher F. Rider, Mohammed O. Altonsy, Mahmoud M. Mostafa, Suharsh V. Shah, Sarah Sasse, Martijn L. Manson, Dong Yan, Carina Kärrman-Mårdh, Anna Miller-Larsson, Anthony N. Gerber, Mark A. Giembycz and Robert NewtonMolecular Pharmacology September 2018, 94 (3) 1031-1046; DOI: https://doi.org/10.1124/mol.118.112755
H
Harrington, Anthony W.
- Open AccessThe Zinc Transporter SLC39A7 (ZIP7) Is Essential for Regulation of Cytosolic Zinc LevelsGrace Woodruff, Christian G. Bouwkamp, Femke M. de Vrij, Timothy Lovenberg, Pascal Bonaventure, Steven A. Kushner and Anthony W. HarringtonMolecular Pharmacology September 2018, 94 (3) 1092-1100; DOI: https://doi.org/10.1124/mol.118.112557
Harvey, Kyle E.
- You have accessMolecular Determinants of the Differential Modulation of Cav1.2 and Cav1.3 by Nifedipine and FPL 64176Yuchen Wang, Shiqi Tang, Kyle E. Harvey, Amy E. Salyer, T. August Li, Emily K. Rantz, Markus A. Lill and Gregory H. HockermanMolecular Pharmacology September 2018, 94 (3) 973-983; DOI: https://doi.org/10.1124/mol.118.112441
Hayes, Michael P.
- You have accessA Novel CRISPR/Cas9-Based Cellular Model to Explore Adenylyl Cyclase and cAMP SignalingMonica Soto-Velasquez, Michael P. Hayes, Aktan Alpsoy, Emily C. Dykhuizen and Val J. WattsMolecular Pharmacology September 2018, 94 (3) 963-972; DOI: https://doi.org/10.1124/mol.118.111849
Hirota, Takeshi
- You have accessNucleosome Positioning and Gene Regulation of the SGLT2 Gene in the Renal Proximal Tubular Epithelial CellsHiroaki Takesue, Takeshi Hirota, Mami Tachimura, Ayane Tokashiki and Ichiro IeiriMolecular Pharmacology September 2018, 94 (3) 953-962; DOI: https://doi.org/10.1124/mol.118.111807
Hockerman, Gregory H.
- You have accessMolecular Determinants of the Differential Modulation of Cav1.2 and Cav1.3 by Nifedipine and FPL 64176Yuchen Wang, Shiqi Tang, Kyle E. Harvey, Amy E. Salyer, T. August Li, Emily K. Rantz, Markus A. Lill and Gregory H. HockermanMolecular Pharmacology September 2018, 94 (3) 973-983; DOI: https://doi.org/10.1124/mol.118.112441
Hu, Dong Gui
- You have accessIntergenic Splicing between Four Adjacent UGT Genes (2B15, 2B29P2, 2B17, 2B29P1) Gives Rise to Variant UGT Proteins That Inhibit Glucuronidation via Protein-Protein InteractionsDong Gui Hu, Julie-Ann Hulin, Dhilushi D. Wijayakumara, Ross A. McKinnon, Peter I. Mackenzie and Robyn MeechMolecular Pharmacology September 2018, 94 (3) 938-952; DOI: https://doi.org/10.1124/mol.118.111773
Hulin, Julie-Ann
- You have accessIntergenic Splicing between Four Adjacent UGT Genes (2B15, 2B29P2, 2B17, 2B29P1) Gives Rise to Variant UGT Proteins That Inhibit Glucuronidation via Protein-Protein InteractionsDong Gui Hu, Julie-Ann Hulin, Dhilushi D. Wijayakumara, Ross A. McKinnon, Peter I. Mackenzie and Robyn MeechMolecular Pharmacology September 2018, 94 (3) 938-952; DOI: https://doi.org/10.1124/mol.118.111773
I
Ieiri, Ichiro
- You have accessNucleosome Positioning and Gene Regulation of the SGLT2 Gene in the Renal Proximal Tubular Epithelial CellsHiroaki Takesue, Takeshi Hirota, Mami Tachimura, Ayane Tokashiki and Ichiro IeiriMolecular Pharmacology September 2018, 94 (3) 953-962; DOI: https://doi.org/10.1124/mol.118.111807
J
Jackson, Robert
- You have accessSmall-Molecule G Protein–Coupled Receptor Kinase Inhibitors Attenuate G Protein–Coupled Receptor Kinase 2–Mediated Desensitization of Vasoconstrictor-Induced Arterial ContractionsRichard D. Rainbow, Sean Brennan, Robert Jackson, Alison J. Beech, Amal Bengreed, Helen V. Waldschmidt, John J. G. Tesmer, R. A. John Challiss and Jonathon M. WilletsMolecular Pharmacology September 2018, 94 (3) 1079-1091; DOI: https://doi.org/10.1124/mol.118.112524
Jurcakova, Danica
- You have accessVoltage-Gated Sodium Channels Regulating Action Potential Generation in Itch-, Nociceptive-, and Low-Threshold Mechanosensitive Cutaneous C-FibersDanica Jurcakova, Fei Ru, Marian Kollarik, Hui Sun, Jeffrey Krajewski and Bradley J. UndemMolecular Pharmacology September 2018, 94 (3) 1047-1056; DOI: https://doi.org/10.1124/mol.118.112839
K
Kärrman-Mårdh, Carina
- You have accessLong-Acting β2-Adrenoceptor Agonists Enhance Glucocorticoid Receptor (GR)–Mediated Transcription by Gene-Specific Mechanisms Rather Than Generic Effects via GRChristopher F. Rider, Mohammed O. Altonsy, Mahmoud M. Mostafa, Suharsh V. Shah, Sarah Sasse, Martijn L. Manson, Dong Yan, Carina Kärrman-Mårdh, Anna Miller-Larsson, Anthony N. Gerber, Mark A. Giembycz and Robert NewtonMolecular Pharmacology September 2018, 94 (3) 1031-1046; DOI: https://doi.org/10.1124/mol.118.112755
Kenakin, Terry
- You have accessEquilibrium Assays Are Required to Accurately Characterize the Activity Profiles of Drugs Modulating Gq-Protein-Coupled ReceptorsSara Bdioui, Julien Verdi, Nicolas Pierre, Eric Trinquet, Thomas Roux and Terry KenakinMolecular Pharmacology September 2018, 94 (3) 992-1006; DOI: https://doi.org/10.1124/mol.118.112573
Kollarik, Marian
- You have accessVoltage-Gated Sodium Channels Regulating Action Potential Generation in Itch-, Nociceptive-, and Low-Threshold Mechanosensitive Cutaneous C-FibersDanica Jurcakova, Fei Ru, Marian Kollarik, Hui Sun, Jeffrey Krajewski and Bradley J. UndemMolecular Pharmacology September 2018, 94 (3) 1047-1056; DOI: https://doi.org/10.1124/mol.118.112839
Krajewski, Jeffrey
- You have accessVoltage-Gated Sodium Channels Regulating Action Potential Generation in Itch-, Nociceptive-, and Low-Threshold Mechanosensitive Cutaneous C-FibersDanica Jurcakova, Fei Ru, Marian Kollarik, Hui Sun, Jeffrey Krajewski and Bradley J. UndemMolecular Pharmacology September 2018, 94 (3) 1047-1056; DOI: https://doi.org/10.1124/mol.118.112839
Kushner, Steven A.
- Open AccessThe Zinc Transporter SLC39A7 (ZIP7) Is Essential for Regulation of Cytosolic Zinc LevelsGrace Woodruff, Christian G. Bouwkamp, Femke M. de Vrij, Timothy Lovenberg, Pascal Bonaventure, Steven A. Kushner and Anthony W. HarringtonMolecular Pharmacology September 2018, 94 (3) 1092-1100; DOI: https://doi.org/10.1124/mol.118.112557
L
Lau, Miranda
- You have accessChaperone Activity and Dimerization Properties of Hsp90α and Hsp90β in Glucocorticoid Receptor Activation by the Multiprotein Hsp90/Hsp70-Dependent Chaperone MachineryYoshihiro Morishima, Ranjit K. Mehta, Miyako Yoshimura, Miranda Lau, Daniel R. Southworth, Theodore S. Lawrence, William B. Pratt, Mukesh K. Nyati and Yoichi OsawaMolecular Pharmacology September 2018, 94 (3) 984-991; DOI: https://doi.org/10.1124/mol.118.112516
Lawrence, Theodore S.
- You have accessChaperone Activity and Dimerization Properties of Hsp90α and Hsp90β in Glucocorticoid Receptor Activation by the Multiprotein Hsp90/Hsp70-Dependent Chaperone MachineryYoshihiro Morishima, Ranjit K. Mehta, Miyako Yoshimura, Miranda Lau, Daniel R. Southworth, Theodore S. Lawrence, William B. Pratt, Mukesh K. Nyati and Yoichi OsawaMolecular Pharmacology September 2018, 94 (3) 984-991; DOI: https://doi.org/10.1124/mol.118.112516
Li, T. August
- You have accessMolecular Determinants of the Differential Modulation of Cav1.2 and Cav1.3 by Nifedipine and FPL 64176Yuchen Wang, Shiqi Tang, Kyle E. Harvey, Amy E. Salyer, T. August Li, Emily K. Rantz, Markus A. Lill and Gregory H. HockermanMolecular Pharmacology September 2018, 94 (3) 973-983; DOI: https://doi.org/10.1124/mol.118.112441
Lill, Markus A.
- You have accessMolecular Determinants of the Differential Modulation of Cav1.2 and Cav1.3 by Nifedipine and FPL 64176Yuchen Wang, Shiqi Tang, Kyle E. Harvey, Amy E. Salyer, T. August Li, Emily K. Rantz, Markus A. Lill and Gregory H. HockermanMolecular Pharmacology September 2018, 94 (3) 973-983; DOI: https://doi.org/10.1124/mol.118.112441
Lovenberg, Timothy
- Open AccessThe Zinc Transporter SLC39A7 (ZIP7) Is Essential for Regulation of Cytosolic Zinc LevelsGrace Woodruff, Christian G. Bouwkamp, Femke M. de Vrij, Timothy Lovenberg, Pascal Bonaventure, Steven A. Kushner and Anthony W. HarringtonMolecular Pharmacology September 2018, 94 (3) 1092-1100; DOI: https://doi.org/10.1124/mol.118.112557
M
Mackenzie, Peter I.
- You have accessIntergenic Splicing between Four Adjacent UGT Genes (2B15, 2B29P2, 2B17, 2B29P1) Gives Rise to Variant UGT Proteins That Inhibit Glucuronidation via Protein-Protein InteractionsDong Gui Hu, Julie-Ann Hulin, Dhilushi D. Wijayakumara, Ross A. McKinnon, Peter I. Mackenzie and Robyn MeechMolecular Pharmacology September 2018, 94 (3) 938-952; DOI: https://doi.org/10.1124/mol.118.111773
Manson, Martijn L.
- You have accessLong-Acting β2-Adrenoceptor Agonists Enhance Glucocorticoid Receptor (GR)–Mediated Transcription by Gene-Specific Mechanisms Rather Than Generic Effects via GRChristopher F. Rider, Mohammed O. Altonsy, Mahmoud M. Mostafa, Suharsh V. Shah, Sarah Sasse, Martijn L. Manson, Dong Yan, Carina Kärrman-Mårdh, Anna Miller-Larsson, Anthony N. Gerber, Mark A. Giembycz and Robert NewtonMolecular Pharmacology September 2018, 94 (3) 1031-1046; DOI: https://doi.org/10.1124/mol.118.112755
McKinnon, Ross A.
- You have accessIntergenic Splicing between Four Adjacent UGT Genes (2B15, 2B29P2, 2B17, 2B29P1) Gives Rise to Variant UGT Proteins That Inhibit Glucuronidation via Protein-Protein InteractionsDong Gui Hu, Julie-Ann Hulin, Dhilushi D. Wijayakumara, Ross A. McKinnon, Peter I. Mackenzie and Robyn MeechMolecular Pharmacology September 2018, 94 (3) 938-952; DOI: https://doi.org/10.1124/mol.118.111773
Meech, Robyn
- You have accessIntergenic Splicing between Four Adjacent UGT Genes (2B15, 2B29P2, 2B17, 2B29P1) Gives Rise to Variant UGT Proteins That Inhibit Glucuronidation via Protein-Protein InteractionsDong Gui Hu, Julie-Ann Hulin, Dhilushi D. Wijayakumara, Ross A. McKinnon, Peter I. Mackenzie and Robyn MeechMolecular Pharmacology September 2018, 94 (3) 938-952; DOI: https://doi.org/10.1124/mol.118.111773
Mehta, Ranjit K.
- You have accessChaperone Activity and Dimerization Properties of Hsp90α and Hsp90β in Glucocorticoid Receptor Activation by the Multiprotein Hsp90/Hsp70-Dependent Chaperone MachineryYoshihiro Morishima, Ranjit K. Mehta, Miyako Yoshimura, Miranda Lau, Daniel R. Southworth, Theodore S. Lawrence, William B. Pratt, Mukesh K. Nyati and Yoichi OsawaMolecular Pharmacology September 2018, 94 (3) 984-991; DOI: https://doi.org/10.1124/mol.118.112516
Miller-Larsson, Anna
- You have accessLong-Acting β2-Adrenoceptor Agonists Enhance Glucocorticoid Receptor (GR)–Mediated Transcription by Gene-Specific Mechanisms Rather Than Generic Effects via GRChristopher F. Rider, Mohammed O. Altonsy, Mahmoud M. Mostafa, Suharsh V. Shah, Sarah Sasse, Martijn L. Manson, Dong Yan, Carina Kärrman-Mårdh, Anna Miller-Larsson, Anthony N. Gerber, Mark A. Giembycz and Robert NewtonMolecular Pharmacology September 2018, 94 (3) 1031-1046; DOI: https://doi.org/10.1124/mol.118.112755
Morishima, Yoshihiro
- You have accessChaperone Activity and Dimerization Properties of Hsp90α and Hsp90β in Glucocorticoid Receptor Activation by the Multiprotein Hsp90/Hsp70-Dependent Chaperone MachineryYoshihiro Morishima, Ranjit K. Mehta, Miyako Yoshimura, Miranda Lau, Daniel R. Southworth, Theodore S. Lawrence, William B. Pratt, Mukesh K. Nyati and Yoichi OsawaMolecular Pharmacology September 2018, 94 (3) 984-991; DOI: https://doi.org/10.1124/mol.118.112516
Mostafa, Mahmoud M.
- You have accessLong-Acting β2-Adrenoceptor Agonists Enhance Glucocorticoid Receptor (GR)–Mediated Transcription by Gene-Specific Mechanisms Rather Than Generic Effects via GRChristopher F. Rider, Mohammed O. Altonsy, Mahmoud M. Mostafa, Suharsh V. Shah, Sarah Sasse, Martijn L. Manson, Dong Yan, Carina Kärrman-Mårdh, Anna Miller-Larsson, Anthony N. Gerber, Mark A. Giembycz and Robert NewtonMolecular Pharmacology September 2018, 94 (3) 1031-1046; DOI: https://doi.org/10.1124/mol.118.112755
N
Newton, Gary K.
- Open AccessAllergen Delivery Inhibitors: A Rationale for Targeting Sentinel Innate Immune Signaling of Group 1 House Dust Mite Allergens through Structure-Based Protease Inhibitor DesignJihui Zhang, Jie Chen, Gary K. Newton, Trevor R. Perrior and Clive RobinsonMolecular Pharmacology September 2018, 94 (3) 1007-1030; DOI: https://doi.org/10.1124/mol.118.112730
Newton, Robert
- You have accessLong-Acting β2-Adrenoceptor Agonists Enhance Glucocorticoid Receptor (GR)–Mediated Transcription by Gene-Specific Mechanisms Rather Than Generic Effects via GRChristopher F. Rider, Mohammed O. Altonsy, Mahmoud M. Mostafa, Suharsh V. Shah, Sarah Sasse, Martijn L. Manson, Dong Yan, Carina Kärrman-Mårdh, Anna Miller-Larsson, Anthony N. Gerber, Mark A. Giembycz and Robert NewtonMolecular Pharmacology September 2018, 94 (3) 1031-1046; DOI: https://doi.org/10.1124/mol.118.112755
Nyati, Mukesh K.
- You have accessChaperone Activity and Dimerization Properties of Hsp90α and Hsp90β in Glucocorticoid Receptor Activation by the Multiprotein Hsp90/Hsp70-Dependent Chaperone MachineryYoshihiro Morishima, Ranjit K. Mehta, Miyako Yoshimura, Miranda Lau, Daniel R. Southworth, Theodore S. Lawrence, William B. Pratt, Mukesh K. Nyati and Yoichi OsawaMolecular Pharmacology September 2018, 94 (3) 984-991; DOI: https://doi.org/10.1124/mol.118.112516
O
Osawa, Yoichi
- You have accessChaperone Activity and Dimerization Properties of Hsp90α and Hsp90β in Glucocorticoid Receptor Activation by the Multiprotein Hsp90/Hsp70-Dependent Chaperone MachineryYoshihiro Morishima, Ranjit K. Mehta, Miyako Yoshimura, Miranda Lau, Daniel R. Southworth, Theodore S. Lawrence, William B. Pratt, Mukesh K. Nyati and Yoichi OsawaMolecular Pharmacology September 2018, 94 (3) 984-991; DOI: https://doi.org/10.1124/mol.118.112516
P
Perrior, Trevor R.
- Open AccessAllergen Delivery Inhibitors: A Rationale for Targeting Sentinel Innate Immune Signaling of Group 1 House Dust Mite Allergens through Structure-Based Protease Inhibitor DesignJihui Zhang, Jie Chen, Gary K. Newton, Trevor R. Perrior and Clive RobinsonMolecular Pharmacology September 2018, 94 (3) 1007-1030; DOI: https://doi.org/10.1124/mol.118.112730
Pierre, Nicolas
- You have accessEquilibrium Assays Are Required to Accurately Characterize the Activity Profiles of Drugs Modulating Gq-Protein-Coupled ReceptorsSara Bdioui, Julien Verdi, Nicolas Pierre, Eric Trinquet, Thomas Roux and Terry KenakinMolecular Pharmacology September 2018, 94 (3) 992-1006; DOI: https://doi.org/10.1124/mol.118.112573
Pratt, William B.
- You have accessChaperone Activity and Dimerization Properties of Hsp90α and Hsp90β in Glucocorticoid Receptor Activation by the Multiprotein Hsp90/Hsp70-Dependent Chaperone MachineryYoshihiro Morishima, Ranjit K. Mehta, Miyako Yoshimura, Miranda Lau, Daniel R. Southworth, Theodore S. Lawrence, William B. Pratt, Mukesh K. Nyati and Yoichi OsawaMolecular Pharmacology September 2018, 94 (3) 984-991; DOI: https://doi.org/10.1124/mol.118.112516
R
Rainbow, Richard D.
- You have accessSmall-Molecule G Protein–Coupled Receptor Kinase Inhibitors Attenuate G Protein–Coupled Receptor Kinase 2–Mediated Desensitization of Vasoconstrictor-Induced Arterial ContractionsRichard D. Rainbow, Sean Brennan, Robert Jackson, Alison J. Beech, Amal Bengreed, Helen V. Waldschmidt, John J. G. Tesmer, R. A. John Challiss and Jonathon M. WilletsMolecular Pharmacology September 2018, 94 (3) 1079-1091; DOI: https://doi.org/10.1124/mol.118.112524
Rantz, Emily K.
- You have accessMolecular Determinants of the Differential Modulation of Cav1.2 and Cav1.3 by Nifedipine and FPL 64176Yuchen Wang, Shiqi Tang, Kyle E. Harvey, Amy E. Salyer, T. August Li, Emily K. Rantz, Markus A. Lill and Gregory H. HockermanMolecular Pharmacology September 2018, 94 (3) 973-983; DOI: https://doi.org/10.1124/mol.118.112441
Rider, Christopher F.
- You have accessLong-Acting β2-Adrenoceptor Agonists Enhance Glucocorticoid Receptor (GR)–Mediated Transcription by Gene-Specific Mechanisms Rather Than Generic Effects via GRChristopher F. Rider, Mohammed O. Altonsy, Mahmoud M. Mostafa, Suharsh V. Shah, Sarah Sasse, Martijn L. Manson, Dong Yan, Carina Kärrman-Mårdh, Anna Miller-Larsson, Anthony N. Gerber, Mark A. Giembycz and Robert NewtonMolecular Pharmacology September 2018, 94 (3) 1031-1046; DOI: https://doi.org/10.1124/mol.118.112755
Robinson, Clive
- Open AccessAllergen Delivery Inhibitors: A Rationale for Targeting Sentinel Innate Immune Signaling of Group 1 House Dust Mite Allergens through Structure-Based Protease Inhibitor DesignJihui Zhang, Jie Chen, Gary K. Newton, Trevor R. Perrior and Clive RobinsonMolecular Pharmacology September 2018, 94 (3) 1007-1030; DOI: https://doi.org/10.1124/mol.118.112730
Rothnie, Alice J.
- You have accessAn Outward-Facing Aromatic Amino Acid Is Crucial for Signaling between the Membrane-Spanning and Nucleotide-Binding Domains of Multidrug Resistance Protein 1 (MRP1; ABCC1)Kevin E. Weigl, Gwenaëlle Conseil, Alice J. Rothnie, May Arama, Yossi Tsfadia and Susan P. C. ColeMolecular Pharmacology September 2018, 94 (3) 1069-1078; DOI: https://doi.org/10.1124/mol.118.112615
Roux, Thomas
- You have accessEquilibrium Assays Are Required to Accurately Characterize the Activity Profiles of Drugs Modulating Gq-Protein-Coupled ReceptorsSara Bdioui, Julien Verdi, Nicolas Pierre, Eric Trinquet, Thomas Roux and Terry KenakinMolecular Pharmacology September 2018, 94 (3) 992-1006; DOI: https://doi.org/10.1124/mol.118.112573
Ru, Fei
- You have accessVoltage-Gated Sodium Channels Regulating Action Potential Generation in Itch-, Nociceptive-, and Low-Threshold Mechanosensitive Cutaneous C-FibersDanica Jurcakova, Fei Ru, Marian Kollarik, Hui Sun, Jeffrey Krajewski and Bradley J. UndemMolecular Pharmacology September 2018, 94 (3) 1047-1056; DOI: https://doi.org/10.1124/mol.118.112839
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Salyer, Amy E.
- You have accessMolecular Determinants of the Differential Modulation of Cav1.2 and Cav1.3 by Nifedipine and FPL 64176Yuchen Wang, Shiqi Tang, Kyle E. Harvey, Amy E. Salyer, T. August Li, Emily K. Rantz, Markus A. Lill and Gregory H. HockermanMolecular Pharmacology September 2018, 94 (3) 973-983; DOI: https://doi.org/10.1124/mol.118.112441
Sandoval, Philip J.
- You have accessAssessment of Substrate-Dependent Ligand Interactions at the Organic Cation Transporter OCT2 Using Six Model SubstratesPhilip J. Sandoval, Kimberley M. Zorn, Alex M. Clark, Sean Ekins and Stephen H. WrightMolecular Pharmacology September 2018, 94 (3) 1057-1068; DOI: https://doi.org/10.1124/mol.117.111443
Sasse, Sarah
- You have accessLong-Acting β2-Adrenoceptor Agonists Enhance Glucocorticoid Receptor (GR)–Mediated Transcription by Gene-Specific Mechanisms Rather Than Generic Effects via GRChristopher F. Rider, Mohammed O. Altonsy, Mahmoud M. Mostafa, Suharsh V. Shah, Sarah Sasse, Martijn L. Manson, Dong Yan, Carina Kärrman-Mårdh, Anna Miller-Larsson, Anthony N. Gerber, Mark A. Giembycz and Robert NewtonMolecular Pharmacology September 2018, 94 (3) 1031-1046; DOI: https://doi.org/10.1124/mol.118.112755
Shah, Suharsh V.
- You have accessLong-Acting β2-Adrenoceptor Agonists Enhance Glucocorticoid Receptor (GR)–Mediated Transcription by Gene-Specific Mechanisms Rather Than Generic Effects via GRChristopher F. Rider, Mohammed O. Altonsy, Mahmoud M. Mostafa, Suharsh V. Shah, Sarah Sasse, Martijn L. Manson, Dong Yan, Carina Kärrman-Mårdh, Anna Miller-Larsson, Anthony N. Gerber, Mark A. Giembycz and Robert NewtonMolecular Pharmacology September 2018, 94 (3) 1031-1046; DOI: https://doi.org/10.1124/mol.118.112755
Soto-Velasquez, Monica
- You have accessA Novel CRISPR/Cas9-Based Cellular Model to Explore Adenylyl Cyclase and cAMP SignalingMonica Soto-Velasquez, Michael P. Hayes, Aktan Alpsoy, Emily C. Dykhuizen and Val J. WattsMolecular Pharmacology September 2018, 94 (3) 963-972; DOI: https://doi.org/10.1124/mol.118.111849
Southworth, Daniel R.
- You have accessChaperone Activity and Dimerization Properties of Hsp90α and Hsp90β in Glucocorticoid Receptor Activation by the Multiprotein Hsp90/Hsp70-Dependent Chaperone MachineryYoshihiro Morishima, Ranjit K. Mehta, Miyako Yoshimura, Miranda Lau, Daniel R. Southworth, Theodore S. Lawrence, William B. Pratt, Mukesh K. Nyati and Yoichi OsawaMolecular Pharmacology September 2018, 94 (3) 984-991; DOI: https://doi.org/10.1124/mol.118.112516
Sun, Hui
- You have accessVoltage-Gated Sodium Channels Regulating Action Potential Generation in Itch-, Nociceptive-, and Low-Threshold Mechanosensitive Cutaneous C-FibersDanica Jurcakova, Fei Ru, Marian Kollarik, Hui Sun, Jeffrey Krajewski and Bradley J. UndemMolecular Pharmacology September 2018, 94 (3) 1047-1056; DOI: https://doi.org/10.1124/mol.118.112839
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Tachimura, Mami
- You have accessNucleosome Positioning and Gene Regulation of the SGLT2 Gene in the Renal Proximal Tubular Epithelial CellsHiroaki Takesue, Takeshi Hirota, Mami Tachimura, Ayane Tokashiki and Ichiro IeiriMolecular Pharmacology September 2018, 94 (3) 953-962; DOI: https://doi.org/10.1124/mol.118.111807
Takesue, Hiroaki
- You have accessNucleosome Positioning and Gene Regulation of the SGLT2 Gene in the Renal Proximal Tubular Epithelial CellsHiroaki Takesue, Takeshi Hirota, Mami Tachimura, Ayane Tokashiki and Ichiro IeiriMolecular Pharmacology September 2018, 94 (3) 953-962; DOI: https://doi.org/10.1124/mol.118.111807
Tang, Shiqi
- You have accessMolecular Determinants of the Differential Modulation of Cav1.2 and Cav1.3 by Nifedipine and FPL 64176Yuchen Wang, Shiqi Tang, Kyle E. Harvey, Amy E. Salyer, T. August Li, Emily K. Rantz, Markus A. Lill and Gregory H. HockermanMolecular Pharmacology September 2018, 94 (3) 973-983; DOI: https://doi.org/10.1124/mol.118.112441
Tesmer, John J. G.
- You have accessSmall-Molecule G Protein–Coupled Receptor Kinase Inhibitors Attenuate G Protein–Coupled Receptor Kinase 2–Mediated Desensitization of Vasoconstrictor-Induced Arterial ContractionsRichard D. Rainbow, Sean Brennan, Robert Jackson, Alison J. Beech, Amal Bengreed, Helen V. Waldschmidt, John J. G. Tesmer, R. A. John Challiss and Jonathon M. WilletsMolecular Pharmacology September 2018, 94 (3) 1079-1091; DOI: https://doi.org/10.1124/mol.118.112524
Tokashiki, Ayane
- You have accessNucleosome Positioning and Gene Regulation of the SGLT2 Gene in the Renal Proximal Tubular Epithelial CellsHiroaki Takesue, Takeshi Hirota, Mami Tachimura, Ayane Tokashiki and Ichiro IeiriMolecular Pharmacology September 2018, 94 (3) 953-962; DOI: https://doi.org/10.1124/mol.118.111807
Trinquet, Eric
- You have accessEquilibrium Assays Are Required to Accurately Characterize the Activity Profiles of Drugs Modulating Gq-Protein-Coupled ReceptorsSara Bdioui, Julien Verdi, Nicolas Pierre, Eric Trinquet, Thomas Roux and Terry KenakinMolecular Pharmacology September 2018, 94 (3) 992-1006; DOI: https://doi.org/10.1124/mol.118.112573
Tsfadia, Yossi
- You have accessAn Outward-Facing Aromatic Amino Acid Is Crucial for Signaling between the Membrane-Spanning and Nucleotide-Binding Domains of Multidrug Resistance Protein 1 (MRP1; ABCC1)Kevin E. Weigl, Gwenaëlle Conseil, Alice J. Rothnie, May Arama, Yossi Tsfadia and Susan P. C. ColeMolecular Pharmacology September 2018, 94 (3) 1069-1078; DOI: https://doi.org/10.1124/mol.118.112615
U
Undem, Bradley J.
- You have accessVoltage-Gated Sodium Channels Regulating Action Potential Generation in Itch-, Nociceptive-, and Low-Threshold Mechanosensitive Cutaneous C-FibersDanica Jurcakova, Fei Ru, Marian Kollarik, Hui Sun, Jeffrey Krajewski and Bradley J. UndemMolecular Pharmacology September 2018, 94 (3) 1047-1056; DOI: https://doi.org/10.1124/mol.118.112839
V
Verdi, Julien
- You have accessEquilibrium Assays Are Required to Accurately Characterize the Activity Profiles of Drugs Modulating Gq-Protein-Coupled ReceptorsSara Bdioui, Julien Verdi, Nicolas Pierre, Eric Trinquet, Thomas Roux and Terry KenakinMolecular Pharmacology September 2018, 94 (3) 992-1006; DOI: https://doi.org/10.1124/mol.118.112573
W
Waldschmidt, Helen V.
- You have accessSmall-Molecule G Protein–Coupled Receptor Kinase Inhibitors Attenuate G Protein–Coupled Receptor Kinase 2–Mediated Desensitization of Vasoconstrictor-Induced Arterial ContractionsRichard D. Rainbow, Sean Brennan, Robert Jackson, Alison J. Beech, Amal Bengreed, Helen V. Waldschmidt, John J. G. Tesmer, R. A. John Challiss and Jonathon M. WilletsMolecular Pharmacology September 2018, 94 (3) 1079-1091; DOI: https://doi.org/10.1124/mol.118.112524
Wang, Yuchen
- You have accessMolecular Determinants of the Differential Modulation of Cav1.2 and Cav1.3 by Nifedipine and FPL 64176Yuchen Wang, Shiqi Tang, Kyle E. Harvey, Amy E. Salyer, T. August Li, Emily K. Rantz, Markus A. Lill and Gregory H. HockermanMolecular Pharmacology September 2018, 94 (3) 973-983; DOI: https://doi.org/10.1124/mol.118.112441
Watts, Val J.
- You have accessA Novel CRISPR/Cas9-Based Cellular Model to Explore Adenylyl Cyclase and cAMP SignalingMonica Soto-Velasquez, Michael P. Hayes, Aktan Alpsoy, Emily C. Dykhuizen and Val J. WattsMolecular Pharmacology September 2018, 94 (3) 963-972; DOI: https://doi.org/10.1124/mol.118.111849
Weigl, Kevin E.
- You have accessAn Outward-Facing Aromatic Amino Acid Is Crucial for Signaling between the Membrane-Spanning and Nucleotide-Binding Domains of Multidrug Resistance Protein 1 (MRP1; ABCC1)Kevin E. Weigl, Gwenaëlle Conseil, Alice J. Rothnie, May Arama, Yossi Tsfadia and Susan P. C. ColeMolecular Pharmacology September 2018, 94 (3) 1069-1078; DOI: https://doi.org/10.1124/mol.118.112615
Wijayakumara, Dhilushi D.
- You have accessIntergenic Splicing between Four Adjacent UGT Genes (2B15, 2B29P2, 2B17, 2B29P1) Gives Rise to Variant UGT Proteins That Inhibit Glucuronidation via Protein-Protein InteractionsDong Gui Hu, Julie-Ann Hulin, Dhilushi D. Wijayakumara, Ross A. McKinnon, Peter I. Mackenzie and Robyn MeechMolecular Pharmacology September 2018, 94 (3) 938-952; DOI: https://doi.org/10.1124/mol.118.111773
Willets, Jonathon M.
- You have accessSmall-Molecule G Protein–Coupled Receptor Kinase Inhibitors Attenuate G Protein–Coupled Receptor Kinase 2–Mediated Desensitization of Vasoconstrictor-Induced Arterial ContractionsRichard D. Rainbow, Sean Brennan, Robert Jackson, Alison J. Beech, Amal Bengreed, Helen V. Waldschmidt, John J. G. Tesmer, R. A. John Challiss and Jonathon M. WilletsMolecular Pharmacology September 2018, 94 (3) 1079-1091; DOI: https://doi.org/10.1124/mol.118.112524
Woodruff, Grace
- Open AccessThe Zinc Transporter SLC39A7 (ZIP7) Is Essential for Regulation of Cytosolic Zinc LevelsGrace Woodruff, Christian G. Bouwkamp, Femke M. de Vrij, Timothy Lovenberg, Pascal Bonaventure, Steven A. Kushner and Anthony W. HarringtonMolecular Pharmacology September 2018, 94 (3) 1092-1100; DOI: https://doi.org/10.1124/mol.118.112557
Wright, Stephen H.
- You have accessAssessment of Substrate-Dependent Ligand Interactions at the Organic Cation Transporter OCT2 Using Six Model SubstratesPhilip J. Sandoval, Kimberley M. Zorn, Alex M. Clark, Sean Ekins and Stephen H. WrightMolecular Pharmacology September 2018, 94 (3) 1057-1068; DOI: https://doi.org/10.1124/mol.117.111443
Y
Yan, Dong
- You have accessLong-Acting β2-Adrenoceptor Agonists Enhance Glucocorticoid Receptor (GR)–Mediated Transcription by Gene-Specific Mechanisms Rather Than Generic Effects via GRChristopher F. Rider, Mohammed O. Altonsy, Mahmoud M. Mostafa, Suharsh V. Shah, Sarah Sasse, Martijn L. Manson, Dong Yan, Carina Kärrman-Mårdh, Anna Miller-Larsson, Anthony N. Gerber, Mark A. Giembycz and Robert NewtonMolecular Pharmacology September 2018, 94 (3) 1031-1046; DOI: https://doi.org/10.1124/mol.118.112755
Yoshimura, Miyako
- You have accessChaperone Activity and Dimerization Properties of Hsp90α and Hsp90β in Glucocorticoid Receptor Activation by the Multiprotein Hsp90/Hsp70-Dependent Chaperone MachineryYoshihiro Morishima, Ranjit K. Mehta, Miyako Yoshimura, Miranda Lau, Daniel R. Southworth, Theodore S. Lawrence, William B. Pratt, Mukesh K. Nyati and Yoichi OsawaMolecular Pharmacology September 2018, 94 (3) 984-991; DOI: https://doi.org/10.1124/mol.118.112516
Z
Zhang, Jihui
- Open AccessAllergen Delivery Inhibitors: A Rationale for Targeting Sentinel Innate Immune Signaling of Group 1 House Dust Mite Allergens through Structure-Based Protease Inhibitor DesignJihui Zhang, Jie Chen, Gary K. Newton, Trevor R. Perrior and Clive RobinsonMolecular Pharmacology September 2018, 94 (3) 1007-1030; DOI: https://doi.org/10.1124/mol.118.112730
Zorn, Kimberley M.
- You have accessAssessment of Substrate-Dependent Ligand Interactions at the Organic Cation Transporter OCT2 Using Six Model SubstratesPhilip J. Sandoval, Kimberley M. Zorn, Alex M. Clark, Sean Ekins and Stephen H. WrightMolecular Pharmacology September 2018, 94 (3) 1057-1068; DOI: https://doi.org/10.1124/mol.117.111443
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