Research ArticleArticle
Equilibrium Assays Are Required to Accurately Characterize the Activity Profiles of Drugs Modulating Gq-Protein-Coupled Receptors
Sara Bdioui, Julien Verdi, Nicolas Pierre, Eric Trinquet, Thomas Roux and Terry Kenakin
Molecular Pharmacology September 2018, 94 (3) 992-1006; DOI: https://doi.org/10.1124/mol.118.112573
Sara Bdioui
Cisbio Bioassays, Codolet, France (S.B., J.V., N.P., E.T., T.R.); and Department of Pharmacology, University of North Carolina School of Medicine, Chapel Hill, North Carolina (T.K.)
Julien Verdi
Cisbio Bioassays, Codolet, France (S.B., J.V., N.P., E.T., T.R.); and Department of Pharmacology, University of North Carolina School of Medicine, Chapel Hill, North Carolina (T.K.)
Nicolas Pierre
Cisbio Bioassays, Codolet, France (S.B., J.V., N.P., E.T., T.R.); and Department of Pharmacology, University of North Carolina School of Medicine, Chapel Hill, North Carolina (T.K.)
Eric Trinquet
Cisbio Bioassays, Codolet, France (S.B., J.V., N.P., E.T., T.R.); and Department of Pharmacology, University of North Carolina School of Medicine, Chapel Hill, North Carolina (T.K.)
Thomas Roux
Cisbio Bioassays, Codolet, France (S.B., J.V., N.P., E.T., T.R.); and Department of Pharmacology, University of North Carolina School of Medicine, Chapel Hill, North Carolina (T.K.)
Terry Kenakin
Cisbio Bioassays, Codolet, France (S.B., J.V., N.P., E.T., T.R.); and Department of Pharmacology, University of North Carolina School of Medicine, Chapel Hill, North Carolina (T.K.)
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Functional Assays for Gq-Protein–Activating Receptor Ligands
Sara Bdioui, Julien Verdi, Nicolas Pierre, Eric Trinquet, Thomas Roux and Terry Kenakin
Molecular Pharmacology September 1, 2018, 94 (3) 992-1006; DOI: https://doi.org/10.1124/mol.118.112573
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