Research ArticleArticle
Pharmacological characterization of 1-(5-chloro-6-(trifluoromethoxy)-1H-benzoimidazol-2-yl)-1H-pyrazole-4-carboxylic acid (JNJ-42041935), a potent and selective HIF prolyl hydroxylase (PHD) inhibitor
Terrance D Barrett, Heather L Palomino, Theresa I Theresa I. Brondstetter, Kimon C Kanelakis, Xiaodong Wu, Peter V Haug, Wen Yan, Andy Young, Hong Hua, Juliet C Hart, Da-Thao Tran, Hariharan Venkatesan, Mark D Rosen, Hillary M Peltier, Kia Sepassi, Michele C Rizzolio, Scott D Bembenek, Tara Mirzadegan, Michael H Rabinowitz and Nigel P Shankley
Molecular Pharmacology March 3, 2011, mol.110.070508; DOI: https://doi.org/10.1124/mol.110.070508
Terrance D Barrett
Heather L Palomino
Theresa I Theresa I. Brondstetter
Kimon C Kanelakis
Xiaodong Wu
Peter V Haug
Wen Yan
Andy Young
Hong Hua
Juliet C Hart
Da-Thao Tran
Hariharan Venkatesan
Mark D Rosen
Hillary M Peltier
Kia Sepassi
Michele C Rizzolio
Scott D Bembenek
Tara Mirzadegan
Michael H Rabinowitz
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Research ArticleArticle
Pharmacological characterization of 1-(5-chloro-6-(trifluoromethoxy)-1H-benzoimidazol-2-yl)-1H-pyrazole-4-carboxylic acid (JNJ-42041935), a potent and selective HIF prolyl hydroxylase (PHD) inhibitor
Terrance D Barrett, Heather L Palomino, Theresa I Theresa I. Brondstetter, Kimon C Kanelakis, Xiaodong Wu, Peter V Haug, Wen Yan, Andy Young, Hong Hua, Juliet C Hart, Da-Thao Tran, Hariharan Venkatesan, Mark D Rosen, Hillary M Peltier, Kia Sepassi, Michele C Rizzolio, Scott D Bembenek, Tara Mirzadegan, Michael H Rabinowitz and Nigel P Shankley
Molecular Pharmacology March 3, 2011, mol.110.070508; DOI: https://doi.org/10.1124/mol.110.070508
Research ArticleArticle
Pharmacological characterization of 1-(5-chloro-6-(trifluoromethoxy)-1H-benzoimidazol-2-yl)-1H-pyrazole-4-carboxylic acid (JNJ-42041935), a potent and selective HIF prolyl hydroxylase (PHD) inhibitor
Terrance D Barrett, Heather L Palomino, Theresa I Theresa I. Brondstetter, Kimon C Kanelakis, Xiaodong Wu, Peter V Haug, Wen Yan, Andy Young, Hong Hua, Juliet C Hart, Da-Thao Tran, Hariharan Venkatesan, Mark D Rosen, Hillary M Peltier, Kia Sepassi, Michele C Rizzolio, Scott D Bembenek, Tara Mirzadegan, Michael H Rabinowitz and Nigel P Shankley
Molecular Pharmacology March 3, 2011, mol.110.070508; DOI: https://doi.org/10.1124/mol.110.070508
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