Research ArticleArticle
Targeted degradation of proteins localized in subcellular compartments by hybrid small molecules
Keiichiro Okuhira, Takuji Shoda, Risa Omura, Nobumichi Ohoka, Takayuki Hattori, Norihito Shibata, Yosuke Demizu, Ryo Sugihara, Asato Ichino, Haruka Kawahara, Yukihiro Itoh, Minoru Ishikawa, Yuichi Hashimoto, Masaaki Kurihara, Susumu Itoh, Hiroyuki Saito and Mikihiko Naito
Molecular Pharmacology December 13, 2016, mol.116.105569; DOI: https://doi.org/10.1124/mol.116.105569
Keiichiro Okuhira
1 Institute of Biomedical Sciences, Tokushima University Graduate School;
Takuji Shoda
2 Division of Organic Chemistry, National Institute of Health Sciences;
Risa Omura
1 Institute of Biomedical Sciences, Tokushima University Graduate School;
Nobumichi Ohoka
3 Division of Molecular Target and Gene Therapy Products, National Institute of Health Sciences;
Takayuki Hattori
3 Division of Molecular Target and Gene Therapy Products, National Institute of Health Sciences;
Norihito Shibata
3 Division of Molecular Target and Gene Therapy Products, National Institute of Health Sciences;
Yosuke Demizu
2 Division of Organic Chemistry, National Institute of Health Sciences;
Ryo Sugihara
1 Institute of Biomedical Sciences, Tokushima University Graduate School;
Asato Ichino
1 Institute of Biomedical Sciences, Tokushima University Graduate School;
Haruka Kawahara
1 Institute of Biomedical Sciences, Tokushima University Graduate School;
Yukihiro Itoh
4 Institute of Molecular and Cellular Biosciences, The University of Tokyo;
Minoru Ishikawa
4 Institute of Molecular and Cellular Biosciences, The University of Tokyo;
Yuichi Hashimoto
4 Institute of Molecular and Cellular Biosciences, The University of Tokyo;
Masaaki Kurihara
2 Division of Organic Chemistry, National Institute of Health Sciences;
Susumu Itoh
5 Showa Pharmaceutical University
Hiroyuki Saito
1 Institute of Biomedical Sciences, Tokushima University Graduate School;
Mikihiko Naito
3 Division of Molecular Target and Gene Therapy Products, National Institute of Health Sciences;
Article Figures & Data
Additional Files
Data Supplement
Files in this Data Supplement:
- Supplemental Figures -
Supplementary Figure 1 - cIAP1/cIAP2/XIAP were not involved in the degradation of the nuclear or mitochondria-localized FLAG-CRABP-II proteins
Supplementary Figure 2 - SNIPER(CRABP)-11 did not affect on the mitochondrial membrane integrity
- Supplemental Figures -
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Research ArticleArticle
Targeted degradation of proteins localized in subcellular compartments by hybrid small molecules
Keiichiro Okuhira, Takuji Shoda, Risa Omura, Nobumichi Ohoka, Takayuki Hattori, Norihito Shibata, Yosuke Demizu, Ryo Sugihara, Asato Ichino, Haruka Kawahara, Yukihiro Itoh, Minoru Ishikawa, Yuichi Hashimoto, Masaaki Kurihara, Susumu Itoh, Hiroyuki Saito and Mikihiko Naito
Molecular Pharmacology December 13, 2016, mol.116.105569; DOI: https://doi.org/10.1124/mol.116.105569
Research ArticleArticle
Targeted degradation of proteins localized in subcellular compartments by hybrid small molecules
Keiichiro Okuhira, Takuji Shoda, Risa Omura, Nobumichi Ohoka, Takayuki Hattori, Norihito Shibata, Yosuke Demizu, Ryo Sugihara, Asato Ichino, Haruka Kawahara, Yukihiro Itoh, Minoru Ishikawa, Yuichi Hashimoto, Masaaki Kurihara, Susumu Itoh, Hiroyuki Saito and Mikihiko Naito
Molecular Pharmacology December 13, 2016, mol.116.105569; DOI: https://doi.org/10.1124/mol.116.105569
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