Research ArticleArticle
A novel selective inverse agonist of the CB2 receptor as a radiolabeled tool compound for kinetic binding studies
Andrea Martella, Huub Sijben, Arne Rufer, Juergen Fingerle, Uwe Grether, Christoph Ullmer, Thomas Hartung, Ad IJzerman, Mario van der Stelt and Laura Heitman
Molecular Pharmacology July 26, 2017, mol.117.108605; DOI: https://doi.org/10.1124/mol.117.108605
Andrea Martella
1 Leiden Academic Centre for Drug Research, Leiden University;
Huub Sijben
1 Leiden Academic Centre for Drug Research, Leiden University;
Arne Rufer
2 F. Hoffmann-La Roche Ltd.;
Juergen Fingerle
2 F. Hoffmann-La Roche Ltd.;
Uwe Grether
2 F. Hoffmann-La Roche Ltd.;
Christoph Ullmer
2 F. Hoffmann-La Roche Ltd.;
Thomas Hartung
2 F. Hoffmann-La Roche Ltd.;
Ad IJzerman
1 Leiden Academic Centre for Drug Research, Leiden University;
Mario van der Stelt
3 Leiden Institute of Chemistry, Leiden University
Laura Heitman
1 Leiden Academic Centre for Drug Research, Leiden University;
Article Figures & Data
Additional Files
Data Supplement
- Supplemental Figure -
Filtration binding comparison between [3H]RO6957022 and [3H]CP55,940
- Supplemental Figure -
In this issue
Research ArticleArticle
A novel selective inverse agonist of the CB2 receptor as a radiolabeled tool compound for kinetic binding studies
Andrea Martella, Huub Sijben, Arne Rufer, Juergen Fingerle, Uwe Grether, Christoph Ullmer, Thomas Hartung, Ad IJzerman, Mario van der Stelt and Laura Heitman
Molecular Pharmacology July 26, 2017, mol.117.108605; DOI: https://doi.org/10.1124/mol.117.108605
Research ArticleArticle
A novel selective inverse agonist of the CB2 receptor as a radiolabeled tool compound for kinetic binding studies
Andrea Martella, Huub Sijben, Arne Rufer, Juergen Fingerle, Uwe Grether, Christoph Ullmer, Thomas Hartung, Ad IJzerman, Mario van der Stelt and Laura Heitman
Molecular Pharmacology July 26, 2017, mol.117.108605; DOI: https://doi.org/10.1124/mol.117.108605
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