Mol Pharm -- Table of Contents (51 [2])

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February 1997; 51 (2)   [Index by Author] [Cover Caption]

       Accelerated Communication

       Articles

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Accelerated Communication:

Ichiro Aramori, Junko Zenkoh, Noriyuki Morikawa, Nuala O'Donnell, Masayuki Asano, Kozo Nakamura, Morita Iwami, Hitoshi Kojo, and Yoshitada Notsu: Novel Subtype-Selective Nonpeptide Bradykinin Receptor Antagonists FR167344 and FR173657
Mol Pharmacol 1997 51: 171-176. [Abstract] [Full Text] [PDF]

Larry S. Barak, Stephen S. G. Ferguson, Jie Zhang, Christopher Martenson, Tobias Meyer, and Marc G. Caron: Internal Trafficking and Surface Mobility of a Functionally Intact $beta$ ₂-Adrenergic Receptor-Green Fluorescent Protein Conjugate
Mol Pharmacol 1997 51: 177-184. [Abstract] [Full Text] [PDF]

Articles:

Rammohan V. Rao, Belinda F. Roettger, Elizabeth M. Hadac, and Laurence J. Miller: Roles of Cholecystokinin Receptor Phosphorylation in Agonist-Stimulated Desensitization of Pancreatic Acinar Cells and Receptor-Bearing Chinese Hamster Ovary Cholecystokinin Receptor Cells
Mol Pharmacol 1997 51: 185-192. [Abstract] [Full Text] [PDF]

Edward Kyle, Len Neckers, Chris Takimoto, Gregory Curt, and Raymond Bergan: Genistein-Induced Apoptosis of Prostate Cancer Cells is Preceded by a Specific Decrease in Focal Adhesion Kinase Activity
Mol Pharmacol 1997 51: 193-200. [Abstract] [Full Text] [PDF]

Gregory J. Downing, Bingfang Yan, and Alan M. Poisner: $beta$ -Adrenoceptor Activation-Induced Placental Prorenin Secretion Is Mediated by Increased Renin Messenger RNA and Protein Synthesis
Mol Pharmacol 1997 51: 201-208. [Abstract] [Full Text] [PDF]

Luc Levesque, Nicholas M. Dean, Henri Sasmor, and Stanley T. Crooke: Antisense Oligonucleotides Targeting Human Protein Kinase C- $alpha$ Inhibit Phorbol Ester-Induced Reduction of Bradykinin-Evoked Calcium Mobilization in A549 Cells
Mol Pharmacol 1997 51: 209-216. [Abstract] [Full Text] [PDF]

Zuzana Strakova, Amalendra Kumar, A. John Watson, and Melvyn S. Soloff: A New Linear V_1A Vasopressin Antagonist and Its Use in Characterizing Receptor/G Protein Interactions
Mol Pharmacol 1997 51: 217-224. [Abstract] [Full Text] [PDF]

Sang Geon Kim, Seon Young Nam, Choon Won Kim, Jeong Hee Kim, Chul Koo Cho, and Seong Yul Yoo: Enhancement of Radiation-Inducible Hepatic Glutathione-S-Transferases Ya, Yb1, Yb2, Yc1, and Yc2 Gene Expression by Oltipraz: Possible Role in Radioprotection
Mol Pharmacol 1997 51: 225-233. [Abstract] [Full Text] [PDF]

Zhi-Liang Lu, Carol A. Curtis, Philip G. Jones, Jose Pavia, and Edward C. Hulme: The Role of the Aspartate-Arginine-Tyrosine Triad in the m1 Muscarinic Receptor: Mutations of Aspartate 122 and Tyrosine 124 Decrease Receptor Expression but Do Not Abolish Signaling
Mol Pharmacol 1997 51: 234-241. [Abstract] [Full Text] [PDF]

Georges Némoz, Claudio Sette, and Marco Conti: Selective Activation of Rolipram-Sensitive, cAMP-Specific Phosphodiesterase Isoforms by Phosphatidic Acid
Mol Pharmacol 1997 51: 242-249. [Abstract] [Full Text] [PDF]

Diego Fornasari, Elena Battaglioli, Adriano Flora, Susanna Terzano, and Francesco Clementi: Structural and Functional Characterization of the Human $alpha$ 3 Nicotinic Subunit Gene Promoter
Mol Pharmacol 1997 51: 250-261. [Abstract] [Full Text] [PDF]

Junko Kurokawa, Satomi Adachi-Akahane, and Taku Nagao: 1,5-Benzothiazepine Binding Domain Is Located on the Extracellular Side of the Cardiac L-Type Ca²⁺ Channel
Mol Pharmacol 1997 51: 262-268. [Abstract] [Full Text] [PDF]

Noboru Fujii, Yoshinori Yamashita, Tamio Mizukami, and Hirofumi Nakano: Correlation between the Formation of Cleavable Complex with Topoisomerase I and Growth-Inhibitory Activity for Saintopin-Type Antibiotics
Mol Pharmacol 1997 51: 269-276. [Abstract] [Full Text] [PDF]

Jesús Pintor, Javier Gualix, and M. Teresa Miras-Portugal: Diinosine Polyphosphates, a Group of Dinucleotides with Antagonistic Effects on Diadenosine Polyphosphate Receptor
Mol Pharmacol 1997 51: 277-284. [Abstract] [Full Text] [PDF]

Charbel Massaad, Marc Lombès, Martine Aggerbeck, Marie-Edith Rafestin-Oblin, and Robert Barouki: Cell-Specific, Promoter-Dependent Mineralocorticoid Agonist Activity of Spironolactone
Mol Pharmacol 1997 51: 285-292. [Abstract] [Full Text] [PDF]

Cindy C. Gerhardt, Remko A. Bakker, Gerard J. Piek, Rudi J. Planta, Erno Vreugdenhil, Josée E. Leysen, and Harm Van Heerikhuizen: Molecular Cloning and Pharmacological Characterization of a Molluscan Octopamine Receptor
Mol Pharmacol 1997 51: 293-300. [Abstract] [Full Text] [PDF]

Signe Perlman, Claudio M. Costa-Neto, Ayumi A. Miyakawa, Hans T. Schambye, Siv A. Hjorth, Antonio C. M. Paiva, Ralph A. Rivero, William J. Greenlee, and Thue W. Schwartz: Dual Agonistic and Antagonistic Property of Nonpeptide Angiotensin AT₁ Ligands: Susceptibility to Receptor Mutations
Mol Pharmacol 1997 51: 301-311. [Abstract] [Full Text] [PDF]

E. S. Burstein, T. A. Spalding, and M. R. Brann: Pharmacology of Muscarinic Receptor Subtypes Constitutively Activated by G Proteins
Mol Pharmacol 1997 51: 312-319. [Abstract] [Full Text] [PDF]

V. Gerzanich, A. Kuryatov, R. Anand, and J. Lindstrom: "Orphan" $alpha$ 6 Nicotinic AChR Subunit Can Form a Functional Heteromeric Acetylcholine Receptor
Mol Pharmacol 1997 51: 320-327. [Abstract] [Full Text] [PDF]

Nina C. Saxena, Torben R. Neelands, and Robert L. Macdonald: Contrasting Actions of Lanthanum on Different Recombinant $gamma$ -Aminobutyric Acid Receptor Isoforms Expressed in L929 Fibroblasts
Mol Pharmacol 1997 51: 328-335. [Abstract] [Full Text] [PDF]

Scott C. Harvey, J. Michael Mcintosh, G. Edward Cartier, Floyd N. Maddox, and Charles W. Luetje: Determinants of Specificity for $alpha$ -Conotoxin MII on $alpha$ 3 $beta$ 2 Neuronal Nicotinic Receptors
Mol Pharmacol 1997 51: 336-342. [Abstract] [Full Text] [PDF]

Murat Bastepe and Barrie Ashby: The Long Cytoplasmic Carboxyl Terminus of the Prostaglandin E₂ Receptor EP₄ Subtype Is Essential for Agonist-Induced Desensitization
Mol Pharmacol 1997 51: 343-349. [Abstract] [Full Text] [PDF]

Ho-Sam Ahn, Carolyn Foster, George Boykow, Leyla Arik, April Smith-Torhan, David Hesk, and Meeta Chatterjee: Binding of a Thrombin Receptor Tethered Ligand Analogue to Human Platelet Thrombin Receptor
Mol Pharmacol 1997 51: 350-356. [Abstract] [Full Text] [PDF]

Cover Caption:

About the cover: Stereo view of the proposed interaction between the neuropeptide Y Y₁ receptor and a nonpeptide analog ofthe carboxyl-terminal four amino acids of neuropeptide Y. Thehelices of the human Y₁ receptor are shown in yellow ribbon, andthe side chains of the binding site are shown in yellow. The nonpeptideanalog BIB 3226 is colored by atom type (green, carbon; red, oxygen;blue, nitrogen; white, hydrogen). The model was derived by comparisonof the affinity of neuropeptide Y and BIB 3226 to a large numberof Y₁ receptor mutants expressed in HeLa cells. From Sautel, M.,K. Rudolph, H. Wittneben, H. Herzog, R. Martinez, M. Munoz, W.Eberlein, W. Engel, P. Walker, A. G. Beck-Sickinger. NeuropeptideY and the nonpeptide antagonist BIBP 3226 share an overlappingbinding siteat the human Y1 receptor. Mol. Pharmacol. 50:285-292(1996).