Paul A. Insel

Editor's Note
Mol Pharmacol 2004 65: 1. [Full Text] [PDF]  

Minireview:

Terry Kenakin

Efficacy as a Vector: the Relative Prevalence and Paucity of Inverse Agonism
Mol Pharmacol 2004 65: 2-11. [Abstract] [Full Text] [PDF] Supplemental Table 1  

Perspectives:

Dieter Rosskopf and Karl H. Jakobs

More Hints on Wnts: Gene Profiling by ₂-Adrenergic Receptor-Frizzled Chimeras
Mol Pharmacol 2004 65: 12-14. [Full Text] [PDF]  

Marietta Kaszkin, Karl-Friedrich Beck, Wolfgang Eberhardt, and Josef Pfeilschifter

Unravelling Green Tea's Mechanisms of Action: More Than Meets the Eye
Mol Pharmacol 2004 65: 15-17. [Full Text] [PDF]  

Articles:

Paul A. Insel

Editor's Note
Mol Pharmacol 2004 65: 1. [Full Text] [PDF]  

Adam R. Karpf, Amy W. Lasek, Ted O. Ririe, Adrianne N. Hanks, Douglas Grossman, and David A. Jones

Limited Gene Activation in Tumor and Normal Epithelial Cells Treated with the DNA Methyltransferase Inhibitor 5-Aza-2'-deoxycytidine
Mol Pharmacol 2004 65: 18-27. [Abstract] [Full Text] [PDF]  

Kaleeckal G. Harikumar, Delia I. Pinon, William S. Wessels, Eric S. Dawson, Terry P. Lybrand, Franklyn G. Prendergast, and Laurence J. Miller

Measurement of Intermolecular Distances for the Natural Agonist Peptide Docked at the Cholecystokinin Receptor Expressed in Situ Using Fluorescence Resonance Energy Transfer
Mol Pharmacol 2004 65: 28-35. [Abstract] [Full Text] [PDF]  

Rommel G. Tirona, Brenda F. Leake, Larissa M. Podust, and Richard B. Kim

Identification of Amino Acids in Rat Pregnane X Receptor that Determine Species-Specific Activation
Mol Pharmacol 2004 65: 36-44. [Abstract] [Full Text] [PDF]  

Hong Li, Craig C. Malbon, and Hsien-Yu Wang

Gene Profiling of Frizzled-1 and Frizzled-2 Signaling: Expression of G-Protein-Coupled Receptor Chimeras in Mouse F9 Teratocarcinoma Embryonal Cells
Mol Pharmacol 2004 65: 45-55. [Abstract] [Full Text] [PDF]  

William R. Kem, Vladimir M. Mahnir, Laszlo Prokai, Roger L. Papke, Xuefang Cao, Susan LeFrancois, Kristin Wildeboer, Katalin Prokai-Tatrai, Julia Porter-Papke, and Ferenc Soti

Hydroxy Metabolites of the Alzheimer's Drug Candidate 3-[(2,4-Dimethoxy)Benzylidene]-Anabaseine Dihydrochloride (GTS-21): Their Molecular Properties, Interactions with Brain Nicotinic Receptors, and Brain Penetration
Mol Pharmacol 2004 65: 56-67. [Abstract] [Full Text] [PDF]  

Moez Bali and Myles H. Akabas

Defining the Propofol Binding Site Location on the GABA_A Receptor
Mol Pharmacol 2004 65: 68-76. [Abstract] [Full Text] [PDF]  

Jang-Yang Chang, Chi-Yen Chang, Ching-Chuan Kuo, Li-Tzong Chen, Yung-Shung Wein, and Yueh-Hsiung Kuo

Salvinal, a Novel Microtubule Inhibitor Isolated from Salvia miltiorrhizae Bunge (Danshen), with Antimitotic Activity in Multidrug-Sensitive and -Resistant Human Tumor Cells
Mol Pharmacol 2004 65: 77-84. [Abstract] [Full Text] [PDF]  

Eric Deprez, Sophie Barbe, Macieij Kolaski, Hervé Leh, Fatima Zouhiri, Christian Auclair, Jean-Claude Brochon, Marc Le Bret, and Jean-François Mouscadet

Mechanism of HIV-1 Integrase Inhibition by Styrylquinoline Derivatives in Vitro
Mol Pharmacol 2004 65: 85-98. [Abstract] [Full Text] [PDF]  

Huei-Wen Chen, Sung-Liang Yu, Jeremy J. W. Chen, Han-Ni Li, Yi-Chen Lin, Pei-Li Yao, Han-Yi Chou, Chiang-Ting Chien, Wen-Jone Chen, Yuan-Teh Lee, and Pan-Chyr Yang

Anti-Invasive Gene Expression Profile of Curcumin in Lung Adenocarcinoma Based on a High Throughput Microarray Analysis
Mol Pharmacol 2004 65: 99-110. [Abstract] [Full Text] [PDF]  

Elisa Tedeschi, Marta Menegazzi, Ying Yao, Hisanori Suzuki, Ulrich Förstermann, and Hartmut Kleinert

Green Tea Inhibits Human Inducible Nitric-Oxide Synthase Expression by Down-Regulating Signal Transducer and Activator of Transcription-1 Activation
Mol Pharmacol 2004 65: 111-120. [Abstract] [Full Text] [PDF]  

Anthone W. Dunah, Ana C. Sirianni, Allen A. Fienberg, Elena Bastia, Michael A. Schwarzschild, and David. G. Standaert

Dopamine D1-Dependent Trafficking of Striatal N-Methyl-D-aspartate Glutamate Receptors Requires Fyn Protein Tyrosine Kinase but Not DARPP-32
Mol Pharmacol 2004 65: 121-129. [Abstract] [Full Text] [PDF]  

Pengfei Gong, Arthur I. Cederbaum, and Natalia Nieto

The Liver-Selective Nitric Oxide Donor O²-Vinyl 1-(pyrrolidin-1-yl)diazen-1-ium-1,2-diolate (V-PYRRO/NO) Protects HepG2 Cells against Cytochrome P450 2E1-Dependent Toxicity
Mol Pharmacol 2004 65: 130-138. [Abstract] [Full Text] [PDF]  

Jennifer A. Calvert and Richard J. Evans

Heterogeneity of P2X Receptors in Sympathetic Neurons: Contribution of Neuronal P2X₁ Receptors Revealed Using Knockout Mice
Mol Pharmacol 2004 65: 139-148. [Abstract] [Full Text] [PDF]  

Bahjat Al-Ani, Kristina K. Hansen, and Morley D. Hollenberg

Proteinase-Activated Receptor-2: Key Role of Amino-Terminal Dipeptide Residues of the Tethered Ligand for Receptor Activation
Mol Pharmacol 2004 65: 149-156. [Abstract] [Full Text] [PDF]  

Nansheng Chen, Bo Li, Timothy H. Murphy, and Lynn A. Raymond

Site within N-Methyl-D-aspartate Receptor Pore Modulates Channel Gating
Mol Pharmacol 2004 65: 157-164. [Abstract] [Full Text] [PDF]  

Jane Sohn Thomsen, Silke Kietz, Anders Ström, and Jan-Åke Gustafsson

HES-1, a Novel Target Gene for the Aryl Hydrocarbon Receptor
Mol Pharmacol 2004 65: 165-171. [Abstract] [Full Text] [PDF]  

Daniel Bauer, Nils Wolfram, Georg F. Kahl, and Karen I. Hirsch-Ernst

Transcriptional Regulation of CYP2B1 Induction in Primary Rat Hepatocyte Cultures: Repression by Epidermal Growth Factor Is Mediated via a Distal Enhancer Region
Mol Pharmacol 2004 65: 172-180. [Abstract] [Full Text] [PDF]  

J. C. Kwok and D. R. Richardson

Examination of the Mechanism(s) Involved in Doxorubicin-Mediated Iron Accumulation in Ferritin: Studies Using Metabolic Inhibitors, Protein Synthesis Inhibitors, and Lysosomotropic Agents
Mol Pharmacol 2004 65: 181-195. [Abstract] [Full Text] [PDF]  

Tuan M. Tran, Jackie Friedman, Eyad Qunaibi, Faiza Baameur, Robert H. Moore, and Richard B. Clark

Characterization of Agonist Stimulation of cAMP-Dependent Protein Kinase and G Protein-Coupled Receptor Kinase Phosphorylation of the ₂-Adrenergic Receptor Using Phosphoserine-Specific Antibodies
Mol Pharmacol 2004 65: 196-206. [Abstract] [Full Text] [PDF]  

Kenji Kuwasako, Yuan-Ning Cao, Yasuko Nagoshi, Toshihiro Tsuruda, Kazuo Kitamura, and Tanenao Eto

Characterization of the Human Calcitonin Gene-Related Peptide Receptor Subtypes Associated with Receptor Activity-Modifying Proteins
Mol Pharmacol 2004 65: 207-213. [Abstract] [Full Text] [PDF]  

Elena Zaks-Makhina, Yonjung Kim, Elias Aizenman, and Edwin S. Levitan

Novel Neuroprotective K⁺ Channel Inhibitor Identified by High-Throughput Screening in Yeast
Mol Pharmacol 2004 65: 214-219. [Abstract] [Full Text] [PDF]  

Joanna E. Summerscales and P. David Josephy

Human Acetyl CoA:Arylamine N-Acetyltransferase Variants Generated by Random Mutagenesis
Mol Pharmacol 2004 65: 220-226. [Abstract] [Full Text] [PDF]  

William R. Hartman and Patricia Hentosh

The Antileukemia Drug 2-Chloro-2'-deoxyadenosine: An Intrinsic Transcriptional Antagonist
Mol Pharmacol 2004 65: 227-234. [Abstract] [Full Text] [PDF]  

Irina A. Vasilevskaya, Tatiana V. Rakitina, and Peter J. O'Dwyer

Quantitative Effects on c-Jun N-Terminal Protein Kinase Signaling Determine Synergistic Interaction of Cisplatin and 17-Allylamino-17-Demethoxygeldanamycin in Colon Cancer Cell Lines
Mol Pharmacol 2004 65: 235-243. [Abstract] [Full Text] [PDF]  

Joeri Auwerx, Robert Esnouf, Erik De Clercq, and Jan Balzarini

Susceptibility of Feline Immunodeficiency Virus/Human Immunodeficiency Virus Type 1 Reverse Transcriptase Chimeras to Non-Nucleoside RT Inhibitors
Mol Pharmacol 2004 65: 244-251. [Abstract] [Full Text] [PDF]  

Lori McGrew, Raymond D. Price, Elizabeth Hackler, Mike S. S. Chang, and Elaine Sanders-Bush

RNA Editing of the Human Serotonin 5-HT_2C Receptor Disrupts Transactivation of the Small G-Protein RhoA
Mol Pharmacol 2004 65: 252-256. [Abstract] [Full Text] [PDF]  

S. Lazareno, V. Dolezal, A. Popham, and N. J. M. Birdsall

Thiochrome Enhances Acetylcholine Affinity at Muscarinic M₄ Receptors: Receptor Subtype Selectivity via Cooperativity Rather than Affinity
Mol Pharmacol 2004 65: 257-266. [Abstract] [Full Text] [PDF]  

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