Mol Pharm -- Table of Contents (74 [6])

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December 2008; 74 (6) [Index by Author] [Cover Caption]

Articles

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Table of Contents (PDF) | Editorial Board (PDF) | Front Matter (PDF) | Back Matter (PDF) |

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Articles:

Rebecca S. Y. Wong, Veronique Bodart, Markus Metz, Jean Labrecque, Gary Bridger, and Simon P. Fricker: Comparison of the Potential Multiple Binding Modes of Bicyclam, Monocylam, and Noncyclam Small-Molecule CXC Chemokine Receptor 4 Inhibitors
Mol Pharmacol 2008 74: 1485-1495. Published online September 2, 2008; 10.1124/mol.108.049775 [Abstract] [Full Text] [PDF]

Nicole A. Horenstein, Fedra M. Leonik, and Roger L. Papke: Multiple Pharmacophores for the Selective Activation of Nicotinic ${alpha}$ 7-Type Acetylcholine Receptors
Mol Pharmacol 2008 74: 1496-1511. Published online September 2, 2008; 10.1124/mol.108.048892 [Abstract] [Full Text] [PDF]

Denise G. Teotico, Jason J. Bischof, Li Peng, Steven A. Kliewer, and Matthew R. Redinbo: Structural Basis of Human Pregnane X Receptor Activation by the Hops Constituent Colupulone
Mol Pharmacol 2008 74: 1512-1520. Published online September 2, 2008; 10.1124/mol.108.050732 [Abstract] [Full Text] [PDF]

Leonardo A. Parra, Tracy Baust, Salah El Mestikawy, Marisol Quiroz, Beth Hoffman, Jack M. Haflett, Jeffrey K. Yao, and Gonzalo E. Torres: The Orphan Transporter Rxt1/NTT4 (SLC6A17) Functions as a Synaptic Vesicle Amino Acid Transporter Selective for Proline, Glycine, Leucine, and Alanine
Mol Pharmacol 2008 74: 1521-1532. Published online September 3, 2008; 10.1124/mol.108.050005 [Abstract] [Full Text] [PDF]

Burkhard Kleuser, Daniela Malek, Ronald Gust, Heinz H. Pertz, and Henrik Potteck: 17-β-Estradiol Inhibits Transforming Growth Factor-β Signaling and Function in Breast Cancer Cells via Activation of Extracellular Signal-Regulated Kinase through the G Protein-Coupled Receptor 30
Mol Pharmacol 2008 74: 1533-1543. Published online September 3, 2008; 10.1124/mol.108.046854 [Abstract] [Full Text] [PDF]

Kong M. Xiong, Richard E. Peterson, and Warren Heideman: Aryl Hydrocarbon Receptor-Mediated Down-Regulation of Sox9b Causes Jaw Malformation in Zebrafish Embryos
Mol Pharmacol 2008 74: 1544-1553. Published online September 10, 2008; 10.1124/mol.108.050435 [Abstract] [Full Text] [PDF]

Carole Fruchart-Gaillard, Gilles Mourier, Catherine Marquer, Enrico Stura, Nigel J. M. Birdsall, and Denis Servent: Different Interactions between MT7 Toxin and the Human Muscarinic M₁ Receptor in Its Free and N-Methylscopolamine-Occupied States
Mol Pharmacol 2008 74: 1554-1563. Published online September 10, 2008; 10.1124/mol.108.050773 [Abstract] [Full Text] [PDF]

Shih-Ya Hung, Houng-Chi Liou, Kai-Hsiang Kang, Ruey-Meei Wu, Chun-Chiang Wen, and Wen-Mei Fu: Overexpression of Heme Oxygenase-1 Protects Dopaminergic Neurons against 1-Methyl-4-Phenylpyridinium-Induced Neurotoxicity
Mol Pharmacol 2008 74: 1564-1575. Published online September 17, 2008; 10.1124/mol.108.048611 [Abstract] [Full Text] [PDF]

Li Ni-Komatsu, ChunXiang Tong, Guangming Chen, Nelya Brindzei, and Seth J. Orlow: Identification of Quinolines that Inhibit Melanogenesis by Altering Tyrosinase Family Trafficking
Mol Pharmacol 2008 74: 1576-1586. Published online September 18, 2008; 10.1124/mol.108.050633 [Abstract] [Full Text] [PDF]

Tobias Eltze, Rainer Boer, Thomas Wagner, Steffen Weinbrenner, Michelle C. McDonald, Christoph Thiemermann, Alexander Bürkle, and Thomas Klein: Imidazoquinolinone, Imidazopyridine, and Isoquinolindione Derivatives as Novel and Potent Inhibitors of the Poly(ADP-ribose) Polymerase (PARP): A Comparison with Standard PARP Inhibitors
Mol Pharmacol 2008 74: 1587-1598. Published online September 22, 2008; 10.1124/mol.108.048751 [Abstract] [Full Text] [PDF]

Taeweon Lee, Ralf Schwandner, Gayathri Swaminath, Jennifer Weiszmann, Mario Cardozo, Joanne Greenberg, Peter Jaeckel, Hongfei Ge, Yingcai Wang, Xianyun Jiao, Jiwen Liu, Frank Kayser, Hui Tian, and Yang Li: Identification and Functional Characterization of Allosteric Agonists for the G Protein-Coupled Receptor FFA2
Mol Pharmacol 2008 74: 1599-1609. Published online September 25, 2008; 10.1124/mol.108.049536 [Abstract] [Full Text] [PDF]

Toru Hosoi, Miyako Sasaki, Tsuyoshi Miyahara, Chie Hashimoto, Suguru Matsuo, Michiko Yoshii, and Koichiro Ozawa: Endoplasmic Reticulum Stress Induces Leptin Resistance
Mol Pharmacol 2008 74: 1610-1619. Published online August 28, 2008; 10.1124/mol.108.050070 [Abstract] [Full Text] [PDF]

Christelle Marminon, Fabrice Anizon, Pascale Moreau, Bruno Pfeiffer, Alain Pierré, Roy M. Golsteyn, Paul Peixoto, Marie-Paule Hildebrand, Marie-Hélène David-Cordonnier, Olivier Lozach, Laurent Meijer, and Michelle Prudhomme: Rebeccamycin Derivatives as Dual DNA-Damaging Agents and Potent Checkpoint Kinase 1 Inhibitors
Mol Pharmacol 2008 74: 1620-1629. Published online September 2, 2008; 10.1124/mol.108.049346 [Abstract] [Full Text] [PDF]

Alice Rothnie, Gwenaëlle Conseil, Andrea Y. T. Lau, Roger G. Deeley, and Susan P. C. Cole: Mechanistic Differences between GSH Transport by Multidrug Resistance Protein 1 (MRP1/ABCC1) and GSH Modulation of MRP1-Mediated Transport
Mol Pharmacol 2008 74: 1630-1640. Published online September 2, 2008; 10.1124/mol.108.049080 [Abstract] [Full Text] [PDF] [Data Supplement]

R. Salas, A. Main, D. A. Gangitano, G. Zimmerman, S. Ben-Ari, H. Soreq, and M. De Biasi: Nicotine Relieves Anxiogenic-Like Behavior in Mice that Overexpress the Read-Through Variant of Acetylcholinesterase but Not in Wild-Type Mice
Mol Pharmacol 2008 74: 1641-1648. Published online September 5, 2008; 10.1124/mol.108.048454 [Abstract] [Full Text] [PDF] [Data Supplement]

Christopher. R. Chiaro, Rushang D. Patel, and Gary. H. Perdew: 12(R)-Hydroxy-5(Z),8(Z),10(E),14(Z)-eicosatetraenoic Acid [12(R)-HETE], an Arachidonic Acid Derivative, Is an Activator of the Aryl Hydrocarbon Receptor
Mol Pharmacol 2008 74: 1649-1656. Published online September 8, 2008; 10.1124/mol.108.049379 [Abstract] [Full Text] [PDF] [Data Supplement]

Chao Yan, Jadwiga K. Kepa, David Siegel, Ian J. Stratford, and David Ross: Dissecting the Role of Multiple Reductases in Bioactivation and Cytotoxicity of the Antitumor Agent 2,5-Diaziridinyl-3-(hydroxymethyl)-6-methyl-1,4-benzoquinone (RH1)
Mol Pharmacol 2008 74: 1657-1665. Published online September 15, 2008; 10.1124/mol.108.050401 [Abstract] [Full Text] [PDF] [Data Supplement]

Andrés Norambuena, M. Inés Poblete, M. Verónica Donoso, C. Sofía Espinoza, Alfonso González, and J. Pablo Huidobro-Toro: P2Y₁ Receptor Activation Elicits Its Partition out of Membrane Rafts and Its Rapid Internalization from Human Blood Vessels: Implications for Receptor Signaling
Mol Pharmacol 2008 74: 1666-1677. Published online September 17, 2008; 10.1124/mol.108.048496 [Abstract] [Full Text] [PDF]

Iolanda Esposito, Maria Chiara Proto, Patrizia Gazzerro, Chiara Laezza, Claudia Miele, Anna Teresa Alberobello, Vittoria D'Esposito, Francesco Beguinot, Pietro Formisano, and Maurizio Bifulco: The Cannabinoid CB1 Receptor Antagonist Rimonabant Stimulates 2-Deoxyglucose Uptake in Skeletal Muscle Cells by Regulating the Expression of Phosphatidylinositol-3-kinase
Mol Pharmacol 2008 74: 1678-1686. Published online September 18, 2008; 10.1124/mol.108.049205 [Abstract] [Full Text] [PDF]

Deirdre Stewart, Rooma Desai, Qi Cheng, Aiping Liu, and Stuart A. Forman: Tryptophan Mutations at Azi-Etomidate Photo-Incorporation Sites on ${alpha}$ ₁ or β₂ Subunits Enhance GABA_A Receptor Gating and Reduce Etomidate Modulation
Mol Pharmacol 2008 74: 1687-1695. Published online September 19, 2008; 10.1124/mol.108.050500 [Abstract] [Full Text] [PDF]

Sheng-Nan Wu, Hsung Peng, Bing-Shuo Chen, Ya-Jean Wang, Pei-Yu Wu, and Ming-Wei Lin: Potent Activation of Large-Conductance Ca²⁺-Activated K⁺ Channels by the Diphenylurea 1,3-Bis-[2-hydroxy-5-(trifluoromethyl)phenyl]urea (NS1643) in Pituitary Tumor (GH₃) Cells
Mol Pharmacol 2008 74: 1696-1704. Published online September 22, 2008; 10.1124/mol.108.049106 [Abstract] [Full Text] [PDF] [Data Supplement]

Mario Mezler, Wilfried Hornberger, Reinhold Mueller, Martin Schmidt, Willi Amberg, Wilfried Braje, Michael Ochse, Hans Schoemaker, and Berthold Behl: Inhibitors of GlyT1 Affect Glycine Transport via Discrete Binding Sites
Mol Pharmacol 2008 74: 1705-1715. Published online September 24, 2008; 10.1124/mol.108.049312 [Abstract] [Full Text] [PDF] [Erratum]

Yongjun Wang, Pamela M. Rogers, Keith R. Stayrook, Chen Su, Gabor Varga, Qi Shen, Sunil Nagpal, and Thomas P. Burris: The Selective Alzheimer's Disease Indicator-1 Gene (Seladin-1/DHCR24) Is a Liver X Receptor Target Gene
Mol Pharmacol 2008 74: 1716-1721. Published online September 24, 2008; 10.1124/mol.108.048538 [Abstract] [Full Text] [PDF]

Brian B. Hasinoff, Daywin Patel, and Kimberley A. O'Hara: Mechanisms of Myocyte Cytotoxicity Induced by the Multiple Receptor Tyrosine Kinase Inhibitor Sunitinib
Mol Pharmacol 2008 74: 1722-1728. Published online September 24, 2008; 10.1124/mol.108.050104 [Abstract] [Full Text] [PDF]

Cover Caption:

About the cover: Superimposition of ɑ-bitter acids onto colupulone ligand within the colupulone-PXR crystal structure. See the article by Teotico et al. on page 1512 of this issue.