Receptor | Ki | Agonist |
---|---|---|
nm | ||
HA wt | 2.1 ± 0.2 | |
wt (no tag) | 0.9 ± 0.2 | |
D338A | 1.5 ± 0.4 | |
K300A | 1.1 ± 0.3 | |
HA wt | 780 ± 360 | |
D338A | 730 ± 130 | |
K300A | 3800 ± 1200 | |
HA wt | 3.9 ± 1.0 | |
D338A | 2.1 ± 0.6 | |
K300A | 3.3 ± 0.6 | |
HA wt | 570 ± 130 | |
D338A | 430 ± 130 | |
K300A | 1000 ± 410 | |
HA wt | 0.6 ± 0.2 | |
wt (no tag) | 0.5 ± 0.1 | |
D338A | 0.5 ± 0.1 | |
K300A | 0.5 ± 0.1 | |
Ki values were averaged from three independent experiments (± standard error), with the exception of PGE2methyl ester binding to KA300 (five experiments).