Table 1

Activation parameters

SampleV½kn
mV
Kv2.12.1  ± 4.217.4  ± 1.37
PKA mutant2.0  ± 3.116.4  ± 1.26
ΔC187−11.2  ± 6.015.3  ± 1.57
ΔC318−11.8  ± 2.91-a 13.4  ± 1.37
Kv2.1 + AP 0′0.9  ± 3.615.4  ± 1.07
Kv2.1 + AP 30′−25.2  ± 3.11-b 16.5  ± 2.17
ΔC318 + AP 0′−10.7  ± 4.613.0  ± 1.58
ΔC318 + AP 30′−24.4  ± 4.314.8  ± 1.08

V ½ and k values were analyzed as described in Experimental Procedures. Data were expressed as mean ± S.D.

    • 1-a p < 0.05 versus Kv2.1.

    • 1-b p < 0.05 versus + AP 0′.