Baculovirus expression: displacement of radiolabels
| Ligand | Mean pKi | |
|---|---|---|
| [125I]AC512 radiolabel | [125I]hCAL radiolabel | |
| Antagonist | ||
| AC512 | 9.97 ± 0.22 | 9.64 ± 0.17 |
| AC66 | 9.88 ± 0.16 | 9.46 ± 0.23 |
| hCGRP8–37 | 6.19 ± 0.10 | 6.33 ± 0.08 |
| AC413 | 9.24 ± 0.22 | 8.82 ± 0.16 |
| Agonist | ||
| hCAL | 7.74 ± 0.10 | 8.36 ± 0.16 |
| Rat CAL | 7.41 ± 0.12 | 8.3 ± 0.16 |
| Eel CAL | 10.11 ± 0.08 | 10.77 ± 0.02 |
| Porcine CAL | 8.95 ± 0.33 | 9.38 ± 0.20 |
| rCGRP | 6.93 ± 0.12 | 7.3 ± 0.26 |
| rAmylin | 7.45 ± 0.12 | 8.34 ± 0.16 |