Antagonist | Mean pKi | Agonist | Mean pKi |
---|---|---|---|
AC512 | 10.5 ± 0.30 | rAMYLIN | 10.29 ± 0.15 |
(n = 4) | (n = 6) | ||
AC66 | 9.12 ± 0.45 | Rat CAL | 6.0 ± 0.08 |
(n = 5) | (n = 4) | ||
AC413 | 9.77 ± 0.32 | hCAL | 6.2 ± 0.05 |
(n = 5) | (n = 5) | ||
hCGRP8–37 | 8.31 ± 0.37 | rCGRP | 9.81 ± 0.54 |
(n = 5) | (n = 6) | ||
Eel CAL | 10.5 ± 0.3 | ||
(n = 4) |