Table 9
HEK 293 cells (clone 77): displacement of [
125
I]AC512
Ligand
Mean p
K
i
Antagonist
AC512
9.24 ± 0.23
(
n
= 3)
AC66
9.67 ± 0.34
(
n
= 3)
hCGRP
8–37
5.67 ± 0.07
(
n
= 3)
Agonist
hCAL
7.0 ± 0.06
(
n
= 3)
Rat CAL
6.8 ± 0.12
(
n
= 3)
rAmylin
7.38 ± 0.06
(
n
= 3)