Table 1

Ki values of NSAIDs to inhibit [14C]PAH uptake via OAT1

Drugs   Concentration TestedKi
     μm
Naproxen 102
Ibuprofen 103.5
Indomethacin 510
Salicylurate 2511
Oxyphenbutazone 15032
Piroxicam  3052
Salicylate 500341
Acetylsalicylate 250428
Phenacetin1000488
Paracetamol25002099