Ligand | CB1 | CB1V5.46F | CB2 | CB2F5.46V |
---|---|---|---|---|
HU-2103-a | 0.18 ± 0.04 | 0.13 ± 0.05 | 0.19 ± 0.04 | 0.15 ± 0.02 |
CP-559403-a | 2.4 ± 0.8 | 2.7 ± 0.8 | 3.4 ± 1.2 | 2.5 ± 0.4 |
Anandamide3-a | 74.2 ± 17.7 | 94.7 ± 35.5 | 113.4 ± 34.3 | 127.2 ± 47.8 |
WIN55212-23-a | 10.3 ± 2.1 | 0.82 ± 0.22 | 0.52 ± 0.11 | 7.9 ± 1.7 |
Values are presented as mean ± S.E. of three separate experiments.
↵3-a EC50 value in nM.