Ki values for selected trypanocides
| Trypanocide | P1 | n | P2 | n | H2 | n |
|---|---|---|---|---|---|---|
| Melarsoprol | 33.1 ± 0.6 | 3 | 0.54 ± 0.15 | 3 | 10.1 ± 2.6 | 3 |
| Pentamidine | 32.2 ± 3.6 | 3 | 0.43 ± 0.02 | 3 | 24.9 ± 6.5 | 3 |
| Diminazene aceturate | 176 ± 33 | 4 | 2.36 ± 0.46 | 3 | 102 ± 17 | 3 |
Uptake of 20 nM [3H]adenosine and 30 nM [3H]hypoxanthine by T. b. brucei bloodstream forms was performed as described in the legend to Table 1.