CYP2B1 | IC50 | KD |
---|---|---|
μM | ||
WT | 0.26 | 0.28 |
V367L | 0.04 | N.D. |
V363L | 0.09 | N.D. |
V363A | 0.31 | N.D. |
S294T | 0.31 | N.D. |
S294A | 0.4 | N.D. |
L58F-I114F-S294T | 0.4 | 0.57 |
V367A | 6 | 4.1 |
L58F-I114F | 34 | 30.5 |
IC50 values are the means of two independent BROD assays performed in duplicate and KD values were determined as described under Experimental Procedures.
N.D., not determined.