Parameter | Tylosin | Erythromycin | Azithromycin |
---|---|---|---|
K i (nM) | 2950 ± 100 | ||
K i * (nM) | 4.98 ± 0.30 | ||
k 4 (min−1) | 1.36 ± 0.20 | ||
k 5 (min−1 × 10−3) | 2.30 ± 0.30 | ||
K er (nM) | 393 ± 22 | ||
K er * (nM) | 36 ± 3 | ||
K az (nM) | 48 ± 5 | ||
K az * (nM) | 7.1 ± 0.4 | ||
k 6 (min−1) | 0.59 ± 0.09 | 0.086 ± 0.011 | |
k 7(min−1) | 0.060 ± 0.008 | 0.015 ± 0.001 | |
k 4/K i (M−1s−1 × 104) | 0.77 ± 0.11 | ||
k 6/K er (M−1s−1 × 104) | 2.5 ± 0.2 | ||
k 6/K az (M−1s−1 × 104) | 3.0 ± 0.3 |