Drug | Receptor | Holding Potential | IC50 | Figure |
---|---|---|---|---|
mV | μM | |||
QX-314 | α3β4 | −50 | 2.9 ± 1.0 | 2A |
QX-314 | α3β4(6′F10′T) | −50 | 125 ± 25 | 2A |
Tetracaine | α3β4 | −50 | 9.0 ± 1.6 | 4A & 5A |
Tetracaine | α3β4 | −100 | 4.4 ± 0.8 | 5A |
Tetracaine | α3β4(6′F10′T) | −50 | 23 ± 6.2 | 4A & 5B |
Tetracaine | α3β4(6′F10′T) | −100 | 11.4 ± 7.1 | 5B |