Receptor | Antagonist | Max Response | n | EC50 | Figure |
---|---|---|---|---|---|
μM | |||||
α3β4 | None | 13-a | 2.1 ± 0.6 | 68 ± 12 | 2C & 4C |
10 μM QX-314 | 0.59 ± 0.02 | 1.6 ± 0.3 | 98 ± 12 | 2 | |
10 μM tetracaine | 0.59 ± 0.03 | 1.1 ± 0.2 | 82 ± 15 | 4 | |
α3β4(6′F10′T) | None | 13-a | 0.8 ± 0.1 | 72 ± 17 | 2D, 4D, & 5C |
10 μM QX-314 | 0.79 ± 0.08 | 0.8 ± 0.1 | 183 ± 56 | 2D | |
10 μM tetracaine | 1.0 ± 0.2 | 0.9 ± 0.2 | 240 ± 62 | 4D | |
100 μM tetracaine | 0.64 ± 0.05 | 0.9 ± 0.14 | 500 ± 136 | 5C |
↵3-a By definition.