Table 3

Curve fits for Hill equations

ReceptorAntagonistMax ResponsenEC50Figure
μM
α3β4None13-a 2.1  ± 0.668  ± 122C & 4C
10 μM QX-3140.59  ± 0.021.6  ± 0.398  ± 122
10 μM tetracaine0.59  ± 0.031.1  ± 0.282  ± 154
α3β4(6′F10′T) None13-a 0.8  ± 0.172  ± 172D, 4D, & 5C
10 μM QX-3140.79  ± 0.080.8  ± 0.1183  ± 562D
10 μM tetracaine1.0  ± 0.20.9  ± 0.2240  ± 624D
100 μM tetracaine0.64  ± 0.050.9  ± 0.14500  ± 1365C
  • 3-a  By definition.