Table 1

Properties of ω̄-amino fatty acids and ω̄-amino acyl-Ala derivatives by interaction with PEPT2

graphic

Apparent K i values ± S.E.M. were calculated from IC50 values derived by nonlinear regression analysis of data shown in Figs. 1A, 2A, and 3A. Percentages of IGly-Glnwere taken from the recordings of the I-V relationships shown in Figs.1B, 2B, and 3B representing the current evoked by 5 mM concentrations of the tested compound and compared with 5 mM of the dipeptide Gly-Gln at a membrane potential of −100 mV.