IC50 | ||||
---|---|---|---|---|
HIVp66/HIVp51 | HIVp66/FIVp51 | FIVp66/FIVp51 | FIVp66/HIVp51 | |
μg/ml | ||||
NNRTIs | ||||
Nevirapine | 0.305 | 0.42 | >50 | >50 |
Delavirdine | 0.119 | 0.072 | >50 | >50 |
Efavirenz | 0.008 | 0.003 | >50 | >50 |
Emivirine | 0.039 | 0.048 | >50 | >50 |
Capravirine | 0.005 | 0.023 | >50 | >50 |
GW867420X | 0.002 | 0.006 | >50 | >50 |
UC-781 | 0.008 | 0.006 | >50 | >50 |
TSAO-m3T | 0.416 | 1.5 | >50 | >50 |
NRTI | ||||
ddGTP (μM) | 0.073 | 0.107 | 0.52 | 0.56 |
PFA (μM) | 28 | 21 | 147 | 147 |
poly(rC) · oligo(dG12–18) was the template/primer and [2,8-3H]dGTP was the radiolabeled substrate.