Homogenous steroid hormone receptor binding assays with SP500263
| Receptor Assay | SP500263 · HCl | |||
|---|---|---|---|---|
| Concentration | % Inhibition | IC50 | Ki | |
| μM | ||||
| ER-α | 0.01 | 89 | 5.5 nM | 211.5 pM |
| Glucocorticoid | 10 | 0 | N.A. | N.A. |
| Progesterone | 10 | 12 | N.A. | N.A. |
| Androgen | 10 | 0 | N.A. | N.A. |
N.A., not applicable.