Molecule | Observed IC50 | Predicted IC50 |
---|---|---|
μM | ||
Caffeine | >100 | 1800 |
S-mephenytoin | >100 | 4500 |
Tolbutamide | >100 | 290 |
Chlorzoxazone | >100 | 5200 |
Morphine | >100 | 700 |
Alfentanil3-b | 112 | 93 |
Debrisoquine | >100 | 6600 |
Sufentanil3-b | 4.2 | 2700 |
Fexofenadine | >100 | 110 |
Fentanyl3-b | 6.5 | 1300 |
Loperamide3-b | 2.7 | 300 |
CP 690423-a | 2.3 | 69 |
Indinavir | 44 | 100 |
Quinidine3-a | 2.2 | 120 |
Nelfinavir | 1.4 | 240 |
Saquinavir | 6.5 | 100 |
Verapamil3-a | 2.1 | –3-c |
Mibefradil | 1.2 | 160 |
Ketoconazole | 1.2 | 110 |
CP 123793-a | 0.7 | 82 |
CP 1474783-a | 0.14 | 10 |
CP 1147693-a | 0.3 | 40 |
CP 1172273-a | 0.074 | 59 |
CP 1015563-a | 0.6 | 73 |
LY3359793-a | 0.024 | 130 |
CP 1144163-a | 0.036 | 76 |
CP 1003563-a | 0.114 | 69 |