Constant | Tylosin | Clarithromycin | Roxithromycin | Erythromycin | Azithromycin |
---|---|---|---|---|---|
K i(μM) | 3.00 ± 0.03 | ||||
k 4(min−1) | 1.50 ± 0.09 | ||||
k 5(min−1 × 10−3) | 2.50 ± 0.20 | ||||
k A (nM) | 200 ± 16 | 400 ± 29 | 390 ± 16 | 48 ± 5 | |
K (nM) | 8 ± 0.5 | 20 ± 1 | 36.0 ± 1.8 | 7.1 ± 0.4 | |
k 6(min−1) | 1.20 ± 0.13 | 1.20 ± 0.12 | 0.60 ± 0.05 | 0.086 ± 0.011 | |
k 7 (min−1) | 0.050 ± 0.002 | 0.06 ± 0.003 | 0.060 ± 0.003 | 0.015 ± 0.001 | |
k assoc × 104 (M−1s−1) | 10.4 ± 0.8 | 5.2 ± 0.4 | 2.8 ± 0.1 | 3.5 ± 0.5 |