Receptor Expressed in Oocytes | Agonist Concentration | Reference | V50 | Slope Factor |
---|---|---|---|---|
mV | ||||
hB1(n = 13) | 2 μM Bradykinin | Simpson et al. (2000) | −43.0 | −13.4 |
rM1 (n = 16) | 10 μM Carbachol | Wood et al. (1999) | −51.8 | −16.2 |
hP2Y4 (n = 9) | 40 μM UTP | Communi et al. (1996) | −53.4 | −18.8 |
hP2Y1 (n = 13) | 20 μM 2MeS-ADP | O'Grady et al. (1996) | −72.51-150 | −18.5 |
hP2Y11 (n = 15) | 80 μM 2MeS-ATP | Communi et al. (1999) | −73.51-150 | −15.6 |
sP2Y (n = 12) | 20 μM 2MeS-ADP | Dranoff et al. (2000) | −76.01-150 | −17.3 |
hP2Y1334tr (n = 9) | 20 μM 2MeS-ADP | O'Grady et al. (1996) | −50.3 | −7.6 |
hP2Y1342tr (n = 18) | 20 μM 2MeS-ADP | O'Grady et al. (1996) | −49.0 | −10.8 |
hP2Y1342tr + Y1 peptide (n = 8) | 20 μM 2MeS-ADP | O'Grady et al. (1996) | −72.31-150 | −13.7 |
hP2Y1349tr (n = 9) | 20 μM 2MeS-ADP | O'Grady et al. (1996) | −56.7 | −18.5 |
hP2Y1360tr (n = 17) | 20 μM 2MeS-ADP | O'Grady et al. (1996) | −64.41-150 | −23.0 |
hP2Y1369tr (n = 10) | 20 μM 2MeS-ADP | O'Grady et al. (1996) | −71.21-150 | −19.2 |
hB1/Y1 chimera (n = 6) | 2 μM Bradykinin | Simpson et al. (2000) | −66.31-150 | −15.5 |
hB1 + Y1 peptide (n = 7) | 2 μM Bradykinin | Simpson et al. (2000) | −68.01-150 | −12.9 |
↵1-150 Value was significantly different from the hB1-bradykinin receptor value (p < 0.05).