Proteins | EC50 of Ca2+ Mobilization | EC50 of Ileum Contraction | |
---|---|---|---|
PKR1 | PKR2 | ||
nM | nM | ||
PK1 | 2.64 ± 0.294 | 2.66 ± 0.76 | 0.60 |
PK2 | 3.23 ± 1.21 | 3.00 ± 0.76 | 0.56 |
A1MPK1 | >1000 | >1000 | >300 |
MetPK1 | >1000 | >1000 | >300 |
Ala6PK1 | >1000 | >1000 | >300 |
delAPK1 | 444.7 ± 2.1 | >1000 | >300 |
C18SPK1 | >1000 | >1000 | >300 |
C60RPK1 | >1000 | >1000 | >300 |
AVITGA-colipase | >1000 | >1000 | >300 |
AVITGA-DKK4 | >1000 | >1000 | >300 |
Peptide 1 | >1000 | >1000 | >300 |
Peptide 2 | >1000 | >1000 | >300 |
Chimera 12 | 9.7 ± 3.56 | 6.95 ± 3.30 | 0.75 |
Chimera 21 | 17.0 ± 10.6 | 15.0 ± 1.01 | 2.02 |
PK2 insert | 498.6 | >1000 | >300 |