Compounds | IC50 | Ki |
---|---|---|
μM | μM | |
TLCT1 (hCNT1) | ||
5-Fluorouridine | 28 | 22 |
2′-Deoxyuridine | 43 | 33 |
5-Fluoro-2′-deoxyuridine | 34 | 26 |
5-Fluoro-5′-deoxyuridineb | 31 | 24 |
Capecitabine | >1000a | >773 |
ARAC/D2 (hCNT2) | ||
5-Fluorouridine | 41 | 34 |
2′-Deoxyuridine | 47 | 39 |
5-Fluoro-2′-deoxyuridine | 99 | 82 |
5-Fluoro-5′-deoxyuridineb | 500 | 411 |
Capecitabine | >1000a | >821 |