Drug | Target Enzyme | Concentrations Tested |
---|---|---|
μM | ||
AACOCF3 | Phospholipase A2 | 6.25—200 |
D609 | Phosphatidylcholine-specific phospholipase C (mitogen-activated protein kinase) | 2.5—80 |
KN-93 | CaM kinase II | 0.625—20 |
W-7 | CaM kinase II MLC kinase | 3.125—100 |
U0126 | MEK1 and MEK2 (p38, protein kinase B) | 1.56—50 |
LY 294002 | Phosphatidylinositol 3-kinase (casein kinase 2) | 1.56—50 |
Wortmannin | Phosphatidylinositol 3-kinase (myosin light chain kinase, PI4 kinase) | 0.313—50 |