α6* | (non-α6)β2* | |
---|---|---|
pM | ||
K d | ||
125I-Epibatidine | 10.2 (34) | 8.7 (25) |
nM | ||
K i | ||
Cytisine | 1.43 (29) | 0.25 (42) |
Nicotine | 5 (33) | 3.3 (36) |
Acetylcholine | 11.3 (37) | 11.5 (32) |
1,1-Dimethy1-4-phenylpiperazinium | 15.7 (40) | 24 (43) |
Dihydro-β-erythroidine | 1012 (36) | 1000 (25) |
d-Tubocurarine | 700 (36) | 1650 (27) |
α-Conotoxin MII | 1.1 (47) | |
>10,000 | >10,000 |