Compounds | CLtotal | CLbile, p | CLbile, b | fB | Transcellular Transport |
---|---|---|---|---|---|
ml/min/kg | ml/min/kg | ml/min/g of liver | μl/min/mg of protein | ||
E217βG | 42.9 ± 2.5 | 27.8 ± 3.5 | 1.23 ± 0.12 | 0.16 | 19.4 ± 1.3 |
Pravastatin | 35.2 ± 3.2 | 27.5 ± 5.1 | 1.32 ± 0.28 | 1.00 | 9.3 ± 0.4 |
LTC4 | 90.9 ± 9.1 | 24.2 ± 5.6 | 0.96 ± 0.22 | 0.16 | 10.4 ± 1.0 |
BQ123 | 31.4 ± 3.2 | 28.2 ± 4.2 | 1.37 ± 0.21 | 1.00 | 7.4 ± 1.2 |
TLC-S | 37.0 ± 1.5 | 33.7 ± 1.7 | 1.56 ± 0.05 | 0.45 | 28.5 ± 3.7 |
Temocaprilat | 12.5 ± 1.6 | 9.7 ± 1.2 | 0.42 ± 0.05 | 0.10 | 4.0 ± 1.3 |
Methotrexate | 12.7 ± 1.9 | 10.7 ± 1.7 | 0.46 ± 0.07 | 0.94 | 0.9 ± 1.0 |