Cells | Km | Vmax | Vmax/Km |
---|---|---|---|
mM | pmol / min / mg of protein | ||
UGT2B7 | 0.38 ± 0.12 | 8.49 ± 0.20 (8.5) | 22.3 (22.3) |
CYP3A4/UGT2B7 | 3.71 ± 0.68 | 7.23 ± 0.41 (9.47) | 1.9 (2.55) |
CYP1A2/UGT2B7 | 0.48 ± 0.14 | 5.22 ± 0.17 (5.77) | 10.9 (12.0) |
CYP2C9/UGT2B7 | 0.20 ± 0.12 | 4.43 ± 0.16 (4.3) | 22.2 (21.5) |