Inhibitor | PDE4A11 (S2) | PDE4A11 (P2) | PDE4A4B (S2) | PDE4A4B (P2) | PDE4A10 (S2) |
---|---|---|---|---|---|
Rolipram | 0.72 ± 0.08 | 0.66 ± 0.12 | 1.31 ± 0.08 | 0.26 ± 0.09 | 0.064 ± 0.009 |
Ariflo (cilomilast) | 0.034 ± 0.005 | 0.034 ± 0.005 | 0.061 ± 0.007 | 0.059 ± 0.004 | 0.13 ± 0.03 |
Roflumilast | 0.0048 ± 0.0004 | 0.0039 ± 0.0002 | 0.0090 ± 0.0016 | 0.0025 ± 0.0009 | 0.0041 ± 0.0008 |
Denbufylline | 0.25 ± 0.06 | 0.31 ± 0.04 | 0.56 ± 0.30 | 0.46 ± 0.20 | 0.59 ± 0.17 |
Ro 20-1724 | 0.99 ± 0.11 | 0.91 ± 0.07 | 2.93 ± 1.16 | 2.90 ± 0.10 | 1.24 ± 0.07 |