Receptor | pKi S-NF (Ki S-NF) |
---|---|
nM | |
5-HT2B WT | 7.66 ± 0.02 (22) |
A1.35P | 7.81 ± 0.07a (15) |
A1.35S | 7.77 ± 0.07 (17) |
L1.38S | 7.76 ± 0.06 (17) |
I1.39T | 7.84 ± 0.07a (14) |
V1.42I | 7.82 ± 0.09 (15) |
V2.53L | 6.43 ± 0.04a (370) |
V2.53I | 7.45 ± 0.04a (35) |
V2.53A | 5.48 ± 0.08a (3,300) |
L3.29I | 7.65 ± 0.07 (22) |
M5.39V | 6.65 ± 0.06a (220) |
V2.53L, M5.39V | 6.09 ± 0.08abc (810) |
E7.36N | 7.80 ± 0.06 (16) |
S7.45C | 7.65 ± 0.05 (22) |
5-HT2A WT | 5.73 ± 0.04 (1900) |
5 HT2A L2.53V | 5.74 ± 0.04 (1800) |
5-HT2C WT | 6.77 ± 0.05 (170) |
5-HT2C V2.53L | 5.8 ± 0.1a (2000) |