Construct | pKh | High Affinity Site | pK1 | Hill Number |
---|---|---|---|---|
% | ||||
hMOP-Gi1αC351I | 8.71 ± 0.18 | 48 ± 4 | 6.96 ± 0.27 | −0.53 ± 0.02 |
hMOPV169E, V173D-Gi1αC351I | 6.02 ± 0.02* | −0.82 ± 0.05* | ||
hMOP-Gi1αG202A, C351I | 8.68 ± 0.23 | 60 ± 2 | 6.69 ± 0.23 | −0.52 ± 0.02 |
hMOPV169E, V173D-Gi1αC351I + hMOP-Gi1αG202A, C351I | 8.47 ± 0.06 | 40 ± 2 | 6.18 ± 0.07 | −0.34 ± 0.01 |
↵* Significantly different from hMOP-Gi1αC351I, P < 0.05.