Parameter | Value |
---|---|
Two-state dimer receptor modela | |
RTb | 0.509 ± 0.008 pmol/mg protein |
c1 | 1.42 ± 0.18 nM |
c2 | 0.098 ± 0.014 nM2 |
[A]50 | 0.313 nM |
Models in Fig. 7 (1:1 equation) | |
R1 | 0.925 ± 0.019 pmol/mg protein |
K1 | 0.228 ± 0.023 nM |
Two-independent-site receptor modelc | |
R1 | 0.63 ± 0.05 pmol/mg protein |
K1 | 0.100 ± 0.014 nM |
R2 | 0.42 ± 0.04 pmol/mg protein |
K2 | 2.6 ± 0.9 nM |