Kinase Target | IC50 | Inhibition |
---|---|---|
μM | ||
TGFβR1 | 0.0485 | |
TGFβR2 | 22% | |
p38α | 0.854 | |
p38β | 1.92 | |
EGFR kinase | 0.686 | |
p38γ | 0% | |
JNK1 | 0% | |
MAPKAPK2 | 29% | |
MKK6 | 37% | |
ERK2 | 20% | |
PKA | 15% | |
PKC | 0% | |
PKD | 6% | |
CDC2 | 61% | |
CaMKII | 10% |
JNK, c-Jun NH2-terminal kinase; MAPKAPK, mitogen-activated protein kinase-activated protein kinase; MKK, mitogen-activated protein kinase kinase; ERK, extracellular signal-regulated kinase; PKA, protein kinase A; PKC, protein kinase C; PKD, protein kinase D; CaMKII, calmodulin-dependent protein kinase II.