Nucleotide | Ki | ||
---|---|---|---|
VC1:IIC2 + FSK | VC1:IIC2 + FSK + Gαs | ||
nM | nM | ||
MANT nucleotides | |||
MANT-GTP | 110 ± 19 | 11 ± 3.8 | |
MANT-ATP | 130 ± 11 | 14 ± 3.7 | |
MANT-EDA-ATP | 5500 ± 1100 | 6700 ± 890 | |
6-MANT-ATP | 11,000 ± 1900 | 9400 ± 1400 | |
MABA-ATP | 10,000 ± 1500 | 9400 ± 2100 | |
MAHA-ATP | 58,000 ± 12,000 | 100,000 ± 15,000 | |
TNP nucleotides | |||
TNP-ATP | 100 ± 30 | 81 ± 27 | |
TNP-ADP | 2000 ± 660 | 1300 ± 280 | |
TNP-AMP | 21,000 ± 7200 | 17,000 ± 6000 | |
TNP-GTP | 430 ± 130 | 83 ± 22 | |
TNP-GDP | 8100 ± 2900 | 9400 ± 1800 | |
TNP-UTP | 92 ± 9 | 92 ± 36 | |
TNP-CTP | 110 ± 16 | 310 ± 76 |