Compound | Calculated pKi |
---|---|
Glisamuride | 8.8 |
CS 476 | 8.3 |
Glicaramide | 8.1 |
Spc 5002 | 8.0 |
Glisindamide | 7.8 |
Glimepiride | 7.7 |
Gliquidone | 7.5 |
71 5w | 7.5 |
Glisentide | 7.1 |
Glibenclamide | 7.1 |
Glisoxepide | 6.8 |
Glipizide | 6.5 |
Glisolamide | 6.4 |
Gliclazide | 5.9 |
Glicondamide | 5.6 |
Glibornuride | 5.4 |
Acetohexamide | 5.0 |
Metahexamide | 4.8 |
Tolazamide | 4.8 |
Tosifen | 4.7 |
Tolbutamide | 4.0 |
Carbutamide | 3.7 |
Chlorpropamide | 3.7 |