Receptor:G Protein Fusion | D2L Gαi1 | D2L Gαi2 | D2L Gαi3 | D2L Gαo1 | ||||||||
---|---|---|---|---|---|---|---|---|---|---|---|---|
Dopamine | S-(—)-3-PPP | Dopamine | S-(—)-3-PPP | Dopamine | S-(—)-3-PPP | Dopamine | S-(—)-3-PPP | |||||
pKh (±S.E.M.) | 7.12 (0.11) | 7.20 (0.12) | 7.52 (0.13) | 7.67 (0.35) | 8.44 (0.15) | |||||||
pKl (±S.E.M.) | 5.75 (0.08) | 6.27 (0.06) | 5.63 (0.17) | 6.47 (0.11) | 5.58 (0.12) | 6.26 (0.07) | 5.82 (0.18) | 6.24 (0.07) | ||||
%Rh | 44 (7) | 55 (4) | 36 (4) | 29 (4) | 29 (2) | |||||||
pKiGTP (±S.E.M.) | 5.53 (0.01) | 6.23 (0.02) | 5.81 (0.01) | 6.52 (0.11) | 5.50 (0.11) | 6.27 (0.11) | 5.86 (0.07) | 6.3 (0.01) |