Signal peptide | Sequence | CAM741 IC50 | Inhibition at 10 μM |
---|---|---|---|
nM | |||
CCL22 + 10 | MARLQTALLVVLVLLAVALQATEA—GPYGANMEDS | >10,000 | |
CCL2 + 10 | MKVSAALLCLLLIAATFIPQGLA—QPDAINAPVT | >10,000 | 23% |
IL-13 SP + 10 | MALLLTTVIALTCLGGFASP—GPVPPSTALR | >10,000 | 27% |
IFN-γ + 5 | MKYTSYILAFQLCIVLGSLGCYC—QDPYV | >10,000 | 45% |
CCR7 SP + 10 | MDLGKPMKSVLVVALLVIFQVCLC—QDEVTDDYIG | >10,000 | 49% |
E-selectin | MIASQFLSALTLVLLIKESGA— | 9753 ± 1791 | |
IL-12p40 + 3 | MCHQQLVISWFSLVFLASPLVA—IWE | 4313 ± 1381 | |
CXCL8 + 7 | MTSKLAVALLAAFLISAALC—EGAVLPR | 1473 ± 764 | |
ICAM-1 + 5 | MAPSSPRPALPALLVLLGALFPGPGNA—QTSVS | 687 ± 220 | |
VEGF | MNFLLSWVHWSLALLLYLHHAKWSQA— | 125 ± 82 |
|
IL, interleukin; IFN, interferon.