TABLE 4
Activation of S247Fα4β2
*
AChRs in a cell line
Transfected Subunit
Agonist
ACh
Nicotine
Cytisine
DMPP
μ
M
None
No activity
No activity
No activity
No activity
α5
0.079 ± 0.020
0.072 ± 0.009
0.040 ± 0.024
0.272 ± 0.082
β3
0.036 ± 0.006
0.017 ± 0.003
0.0049 ± 0.0004
0.065 ± 0.009