Compound | Properties | Concentration | -Fold Induction |
---|---|---|---|
μM | |||
GW501516 | Synthetic PPARβ/δ agonist | 1.0 | 16.6 ± 6.0* |
L165,041 | Synthetic PPAR/β/δ agonist | 2.0 | 11.2 ± 4.9* |
cPGI | Synthetic PPARβ/δ agonist | 1.0 | 6.7 ± 1.7* |
GW1929 | Synthetic PPARγ agonist | 0.3 | 1.3 ± 0.6** |
Arachidonic acid | Pan-PPAR ligand | 20 | 2.6 ± 1.1* |
Linoleic acid | Pan-PPAR ligand | 20 | 1.6 ± 0.3* |
Eicosapentaenoic acid | Pan-PPAR ligand | 20 | 1.9 ± 0.4* |
atRA | RAR agonist | 1.0 | 1.1 ± 0.1** |
9-cis-RA | RAR and RxR agonist | 1.0 | 1.0 ± 0** |